SCHEMBL8629880

SCHEMBL8629880

COC(=O)c1cccnc1S(N)(=O)=O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.57
CA2 P00918 1/20 0.57
CA5A P35218 1/20 0.57
CA9 Q16790 1/20 0.57
KDM4E B2RXH2 5/20 0.50
TDP1 Q9NUW8 2/20 0.50
MAP2K1 Q02750 1/20 0.48
LMNA P02545 1/20 0.47
TSHR P16473 1/20 0.47
SLC40A1 Q9NP59 1/20 0.46
ALDH1A1 P00352 2/20 0.46
CFTR P13569 1/20 0.46
HSD17B10 Q99714 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
PKM P14618 1/20 0.46
P2RX7 Q99572 1/20 0.45
POLB P06746 3/20 0.45
ATM Q13315 1/20 0.45
CNR2 P34972 1/20 0.43
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29086564 0.85 TDP1 (0.51) CA1CA2CA5ACA9KDM4E
Methyl Alcohol SCHEMBL27853401 0.84 TDP1 (0.50) CA1CA2CA5ACA9KDM4E
SCHEMBL3714382 0.84 TDP1 (0.50) CA1CA2CA5ACA9KDM4E
SCHEMBL9363595 0.81 P2RX7 (0.49) CA1CA2CA9LMNAP2RX7
SCHEMBL5151972 0.80 NAPRT (0.56) CA1CA2CA9KDM4ETDP1
SCHEMBL2213767 0.80 PARP1 (0.51) CA1CA2CA9KDM4ETDP1
SCHEMBL9117916 0.79 SLC40A1 (0.48) CA1CA2CA5ACA9KDM4E
SCHEMBL22010548 0.79 CA1 (0.45) CA1CA2CA5ACA9KDM4E
SCHEMBL1466611 0.78 TDP1 (0.51) CA1CA2CA5ACA9KDM4E
SCHEMBL1248162 0.78 P2RX7 (0.66) CA1CA2CA5ACA9KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1035287-A The neighbour of weeding-methoxycarbonyl sulfonylurea DU PONT (US) 1989-09-06 CN claimed
EP-3986879-B1 FUSED 1,2-THIAZOLES AND 1,2-THIAZINES WHICH ACT AS NLRP3 MODULATORS AC IMMUNE SA (CH) 2024-10-02 EP disclosed
EP-3880666-B1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2023-06-28 EP disclosed
US-20230024859-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2023-01-26 US disclosed
US-20220378801-A1 NOVEL COMPOUNDS AC IMMUNE SA (CH) 2022-12-01 US disclosed
EP-3986879-A1 FUSED 1,2 THIAZOLES AND 1,2 THIAZINES WHICH ACT AS NL3P3 MODULATORS AC Immune SA (CH) 2022-04-27 EP disclosed
CN-114008030-A Fused 1, 2-thiazoles and 1, 2-thiazines as NLRP3 modulators AC免疫有限公司 2022-02-01 CN disclosed
WO-2020102100-A9 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2022-01-06 WO disclosed
WO-2020102100-A9 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2022-01-06 WO disclosed
EP-3880666-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY Novartis AG (CH) 2021-09-22 EP disclosed
WO-2020102100-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS INFLAMMASOME RESEARCH, INC. (US) 2020-05-22 WO disclosed
WO-2020102100-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS INFLAMMASOME RESEARCH, INC. (US) 2020-05-22 WO disclosed
US-5847126-A N-azinyl-N'-(het) arylsulphonyl-ureas BAYER AKTIENGESELLSCHAFT (DE) 1998-12-08 US disclosed
EP-0645386-B1 N-Azinyl-N'-(het)arylsulfonylureas as herbicides BAYER AG (DE) 1997-12-29 EP disclosed
US-5696257-A INTERMEDIATES FOR HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 1997-12-09 US disclosed
EP-0541407-B1 Nitrogen containing bicyclic derivatives, method for their preparation and pharmaceutical compositions containing them ADIR (FR) 1997-02-26 EP disclosed
US-5580842-A HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 1996-12-03 US disclosed
US-5476936-A Herbicides BAYER AKTIENGESELLSCHAFT (DE) 1995-12-19 US disclosed
EP-0645386-A1 N-Azinyl-N'-(het)arylsulfonylureas as herbicides BAYER AG (DE) 1995-03-29 EP disclosed
CN-1035287-A The neighbour of weeding-methoxycarbonyl sulfonylurea DU PONT (US) 1989-09-06 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230024859-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NLRP1, NLRP3, NOD1 CA1 3841/4885CA2 1348/4885CA5A 1703/4885
US-20220378801-A1 NOVEL COMPOUNDS NLRP3, IL1B, IL18 CA1 4311/4885CA2 4210/4885CA5A 2377/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.