SCHEMBL8635252

SCHEMBL8635252

Cc1cc(Nc2cccc(Cl)c2)c(S(C)(=O)=O)cc1C(=O)Cl

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 2/20 0.50
AKR1C2 P52895 2/20 0.50
ADORA3 P0DMS8 1/20 0.46
ADORA2A P29274 1/20 0.46
ADORA2B P29275 1/20 0.46
ADORA1 P30542 1/20 0.46
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
LMNA P02545 2/20 0.44
HPGD P15428 1/20 0.44
GFER P55789 1/20 0.44
PTGS1 P23219 1/20 0.44
PTGS2 P35354 1/20 0.44
IDH1 O75874 1/20 0.41
ALDH1A1 P00352 1/20 0.41
PDE4B Q07343 1/20 0.41
MAPT P10636 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8635463 0.87 AKR1C3 (0.45) AKR1C3AKR1C2MEN1KMT2AGFER
SCHEMBL8632908 0.87 PTGS1 (0.43) MEN1KMT2ASMN1; SMN2LMNAPTGS1
SCHEMBL8631102 0.86 AKR1C3 (0.47) AKR1C3AKR1C2MEN1KMT2ALMNA
SCHEMBL8633209 0.86 MEN1 (0.43) AKR1C3AKR1C2ADORA3ADORA2AADORA2B
SCHEMBL8637536 0.85 AKR1C3 (0.51) AKR1C3AKR1C2MEN1KMT2ASMN1; SMN2
SCHEMBL7764005 0.84 SLC9A1 (0.57)
SCHEMBL8632107 0.84 AKR1C3 (0.52) AKR1C3AKR1C2IDH1
SCHEMBL8634318 0.84 PDE4B (0.46) MEN1KMT2APTGS1PTGS2ALDH1A1
SCHEMBL8635848 0.81 CYP11B2 (0.46) MEN1KMT2ALMNAALDH1A1PDE4B
SCHEMBL8633408 0.80 ALDH1A1 (0.39) SMN1; SMN2PTGS1PTGS2IDH1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1057999-C 4-Aminobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 2000-11-01 CN disclosed
US-5739142-A 4-aminobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-14 US disclosed
CN-1138575-A 4-aminobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 1996-12-25 CN disclosed