SCHEMBL8633168

SCHEMBL8633168

c1ccc2cc(N3CCN(Cn4ncc5ccccc54)CC3)ncc2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.55
RECQL P46063 2/20 0.41
P2RX7 Q99572 1/20 0.41
LRRK2 Q5S007 1/20 0.41
POLB P06746 3/20 0.40
HSD17B10 Q99714 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CXCR3 P49682 1/20 0.39
CYP1A2 P05177 1/20 0.39
KCNH2 Q12809 1/20 0.39
KMO O15229 1/20 0.38
ADRA2A P08913 1/20 0.37
HTR1A P08908 1/20 0.37
DRD2 P14416 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
DRD3 P35462 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
MAPT P10636 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8628179 0.83 KDM4E (0.50) POLBHSD17B10KCNH2HTR1ADRD2
SCHEMBL8628029 0.82 DRD2 (0.46) HTR3ARECQLP2RX7POLBHSD17B10
SCHEMBL8630532 0.82 DRD2 (0.46) RECQLP2RX7POLBHSD17B10L3MBTL1
SCHEMBL8628045 0.82 DHFR (0.43) HTR3ARECQLP2RX7POLBHSD17B10
SCHEMBL8632193 0.80 KDM4E (0.52) LRRK2HSD17B10L3MBTL1CXCR3DRD2
SCHEMBL8627836 0.80 DRD4 (0.45) HTR3ARECQLP2RX7POLBHSD17B10
SCHEMBL8634968 0.80 DRD4 (0.57) POLBHSD17B10L3MBTL1CYP1A2MAPT
SCHEMBL8633681 0.80 RECQL (0.50) RECQLP2RX7POLBHSD17B10L3MBTL1
SCHEMBL8631634 0.80 HRH3 (0.59) HTR3ARECQLHSD17B10CYP1A2HTR1A
Hydrochloric Acid SCHEMBL8629946 0.79 DRD4 (0.56) POLBHSD17B10L3MBTL1CYP1A2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780475-A Antipsychotic indazole derivatives MERCK, SHARP & DOHME LIMITED (GB) 1998-07-14 US disclosed