SCHEMBL8633199

SCHEMBL8633199

CCc1cc(N(C)c2cccc(C#N)c2)c(S(C)(=O)=O)cc1C(=O)Cl

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PER2 O15055 1/20 0.36
CRY1 Q16526 1/20 0.36
CRY2 Q49AN0 1/20 0.36
CNR1 P21554 5/20 0.35
KCNN4 O15554 1/20 0.34
KCNA5 P22460 1/20 0.34
P4HB P07237 5/20 0.34
KCNJ6 P48051 1/20 0.34
KCNJ5 P48544 1/20 0.34
KCNJ3 P48549 1/20 0.34
CNR2 P34972 2/20 0.33
PDCD1 Q15116 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
KDM4C Q9H3R0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634221 0.88 SIRT2 (0.34)
SCHEMBL8635870 0.87 KCNJ6 (0.39) PER2CRY1CRY2CNR1P4HB
SCHEMBL7768615 0.85 SLC9A1 (0.41)
SCHEMBL8633117 0.85 PDE4B (0.40)
SCHEMBL8635203 0.84 HSP90AA1 (0.35)
SCHEMBL8635349 0.84 ALDH1A1 (0.39) PER2
SCHEMBL8635879 0.82 MTNR1A (0.43)
SCHEMBL8636273 0.82 ALDH1A1 (0.36)
SCHEMBL8634504 0.79 FLT1 (0.38)
SCHEMBL8633074 0.79 CYP3A4 (0.37) KCNA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739142-A 4-aminobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-14 US disclosed