SCHEMBL8668032

SCHEMBL8668032

O=C(O)C1Cc2cc(F)c(F)cc2N(C2CC2)C1=O

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
TSHR P16473 1/20 0.33
AGTR2 P50052 1/20 0.31
ALDH1A1 P00352 2/20 0.31
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.31
TOP2A P11388 1/20 0.31
CYP2C9 P11712 1/20 0.31
HPGD P15428 1/20 0.31
TOP2B Q02880 1/20 0.31
HSD17B10 Q99714 1/20 0.31
DUSP3 P51452 1/20 0.31
POLB P06746 1/20 0.30
FFAR4 Q5NUL3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8817061 0.89 HTR2A (0.34) MEN1KMT2AALDH1A1KDM4ECYP1A2
SCHEMBL4909217 0.82 ALDH1A1 (0.31) ALDH1A1
SCHEMBL1985195 0.79 MEN1 (0.31) MEN1KMT2AFFAR4
SCHEMBL6052739 0.77 KEAP1 (0.35) DUSP3
SCHEMBL10485479 0.76 FFAR4 (0.31) FFAR4
SCHEMBL10785290 0.72 MAOA (0.38) TSHRALDH1A1KDM4ELMNACYP1A2
SCHEMBL7024322 0.67 DRD2 (0.33) MEN1KMT2AALDH1A1KDM4EHPGD
SCHEMBL18091502 0.67 KDM4E (0.45) MEN1KMT2AALDH1A1KDM4EHPGD
SCHEMBL8775559 0.66 TOP2A (0.35) TSHRTOP2APOLB
SCHEMBL10558051 0.63 KDM4E (0.36) ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5783708-A HEXAHYDROISOINDOLE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 1998-07-21 US disclosed
US-5391763-A 3-aza-bicyclo[3.1.0]hexanes which are intermediates for anti-bacterial azabicyclo quinolone carboxylic acids PFIZER INC. (US) 1995-02-21 US disclosed
EP-0297858-A2 Bridged-diazabicycloalkyl quinolone carboxylic acids and esters PFIZER INC. (US) 1989-01-04 EP disclosed