SCHEMBL874785

SCHEMBL874785

Nc1ccccc1-c1nc(C(F)(F)C(F)(F)F)c(C(=O)O)s1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 7/20 0.41
KDM4E B2RXH2 6/20 0.41
ALDH1A1 P00352 5/20 0.41
MAPT P10636 5/20 0.41
RAB9A P51151 4/20 0.41
KMT2A Q03164 3/20 0.41
GAA P10253 3/20 0.41
NPC1 O15118 3/20 0.41
TDP1 Q9NUW8 3/20 0.41
MEN1 O00255 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CDC7 O00311 3/20 0.38
DBF4 Q9UBU7 3/20 0.38
CDK2 P24941 2/20 0.38
CCNE1 P24864 1/20 0.38
POLB P06746 1/20 0.35
PPARG P37231 1/20 0.35
NCOA2 Q15596 1/20 0.35
NCOA1 Q15788 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL874117 0.78 RAB9A (0.48) SMN1; SMN2KDM4EALDH1A1MAPTRAB9A
SCHEMBL874301 0.74 ALDH1A1 (0.40) ALDH1A1MAPTRAB9AKMT2ANPC1
SCHEMBL10820841 0.70 ALDH1A1 (0.53) SMN1; SMN2KDM4EALDH1A1MAPTRAB9A
SCHEMBL4497703 0.70 SMN1; SMN2 (0.59) SMN1; SMN2KDM4EALDH1A1MAPTRAB9A
SCHEMBL874267 0.69 ALDH1A1 (0.39) SMN1; SMN2KDM4EALDH1A1RAB9AGAA
SCHEMBL873941 0.67 RAB9A (0.48) SMN1; SMN2KDM4EALDH1A1MAPTRAB9A
SCHEMBL6228168 0.67 ALDH1A1 (0.67) SMN1; SMN2KDM4EALDH1A1MAPTRAB9A
SCHEMBL3436651 0.66 SMN1; SMN2 (0.67) SMN1; SMN2KDM4EALDH1A1MAPTRAB9A
SCHEMBL6249569 0.65 NFKB1 (0.39) SMN1; SMN2KDM4EALDH1A1RAB9ACDC7
SCHEMBL6183496 0.65 ACHE (0.66) KDM4EALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed