SCHEMBL8744696

SCHEMBL8744696

N#Cc1nc(-c2ccccc2Cl)c[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 3/20 0.46
LRRK2 Q5S007 1/20 0.43
ADORA2A P29274 2/20 0.43
ADORA1 P30542 2/20 0.43
GAA P10253 2/20 0.43
IDO1 P14902 1/20 0.42
PSMB8 P28062 1/20 0.41
HPGD P15428 4/20 0.41
KMT2A Q03164 3/20 0.41
LMNA P02545 1/20 0.41
PDGFRB P09619 1/20 0.40
KDM4E B2RXH2 6/20 0.39
ALDH1A1 P00352 6/20 0.39
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
HSD17B10 Q99714 2/20 0.38
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31218523 0.81 TRPA1 (0.40) LRRK2
SCHEMBL8744729 0.81 KDM4E (0.46) GAAPSMB8HPGDKMT2ALMNA
SCHEMBL8744776 0.80 LRRK2 (0.43) LRRK2GAAIDO1HPGDKMT2A
SCHEMBL8744748 0.80 IDO1 (0.41) L3MBTL1GAAIDO1HPGDKMT2A
SCHEMBL25357822 0.78 USP8 (0.38) L3MBTL1LRRK2PSMB8HPGDKMT2A
SCHEMBL8744737 0.76 CTSK (0.47)
SCHEMBL8744697 0.76 TRPA1 (0.37) L3MBTL1ADORA2AGAAKMT2APDGFRB
SCHEMBL7432291 0.75 ADORA2A (0.41) L3MBTL1LRRK2ADORA2AADORA1GAA
SCHEMBL9876453 0.75 ALDH1A1 (0.46) L3MBTL1GAAHPGDKMT2AKDM4E
SCHEMBL8744801 0.74 NUDT1 (0.38) LRRK2ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0653421-B1 Process for preparing 2-cyanoimidazole compounds ISHIHARA SANGYO KAISHA (JP) 1997-01-15 EP disclosed
US-5552557-A Process for preparing 2-cyanoimidazole compounds by reaction of an amino ketone compound ISHIHARA SANGYO KAISHA, LTD. (JP) 1996-09-03 US disclosed
EP-0653421-A1 Process for preparing 2-cyanoimidazole compounds ISHIHARA SANGYO KAISHA LTD. (JP) 1995-05-17 EP disclosed