SCHEMBL8744776

SCHEMBL8744776

Cc1ccccc1-c1c[nH]c(C#N)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.43
IDO1 P14902 1/20 0.41
METAP2 P50579 1/20 0.41
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
LMNA P02545 2/20 0.38
CASP3 P42574 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
TSHR P16473 2/20 0.37
DCUN1D1 Q96GG9 2/20 0.37
KDM5A P29375 1/20 0.36
AR P10275 3/20 0.36
ALDH1A1 P00352 4/20 0.36
HPGD P15428 2/20 0.36
HTT P42858 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
MEN1 O00255 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8744801 0.87 NUDT1 (0.38) LRRK2TSHRARUSP8
SCHEMBL27857839 0.83 IDO1 (0.41) LRRK2IDO1METAP2NPC1RAB9A
SCHEMBL31218523 0.81 TRPA1 (0.40) LRRK2
SCHEMBL8744731 0.81 HSP90AB1 (0.45) NPC1LMNANPSR1MEN1KMT2A
SCHEMBL8744696 0.80 L3MBTL1 (0.46) LRRK2IDO1NPC1RAB9ASMN1; SMN2
SCHEMBL8744748 0.80 IDO1 (0.41) IDO1NPC1RAB9ASMN1; SMN2LMNA
SCHEMBL8699164 0.77 IDO1 (0.44) IDO1METAP2NPC1RAB9ASMN1; SMN2
SCHEMBL8744737 0.76 CTSK (0.47) ARCYP1A2CYP3A4
SCHEMBL7432291 0.75 ADORA2A (0.41) LRRK2RAB9ASMN1; SMN2LMNAALDH1A1
SCHEMBL9876453 0.75 ALDH1A1 (0.46) RAB9ASMN1; SMN2ALDH1A1HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0653421-B1 Process for preparing 2-cyanoimidazole compounds ISHIHARA SANGYO KAISHA (JP) 1997-01-15 EP disclosed
US-5552557-A Process for preparing 2-cyanoimidazole compounds by reaction of an amino ketone compound ISHIHARA SANGYO KAISHA, LTD. (JP) 1996-09-03 US disclosed
EP-0653421-A1 Process for preparing 2-cyanoimidazole compounds ISHIHARA SANGYO KAISHA LTD. (JP) 1995-05-17 EP disclosed