SCHEMBL8744737

SCHEMBL8744737

N#Cc1nc(-c2ccccc2C(F)(F)F)c[nH]1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSK P43235 1/20 0.47
TRPA1 O75762 5/20 0.44
AR P10275 1/20 0.43
ACP1 P24666 3/20 0.41
KMO O15229 2/20 0.40
VCP P55072 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
HSD11B1 P28845 1/20 0.37
C1R P00736 1/20 0.37
SCN9A Q15858 1/20 0.37
TRPM8 Q7Z2W7 1/20 0.37
NOTUM Q6P988 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31218523 0.78 TRPA1 (0.40) TRPA1
SCHEMBL8744696 0.76 L3MBTL1 (0.46)
SCHEMBL8744748 0.76 IDO1 (0.41) C1R
SCHEMBL8744776 0.76 LRRK2 (0.43) ARCYP1A2CYP3A4
SCHEMBL16481863 0.76 HSD11B1 (0.47) CTSKTRPA1ARACP1KMO
SCHEMBL9870039 0.73 KMO (0.40) CTSKTRPA1ACP1KMOCYP1A2
SCHEMBL7432291 0.72 ADORA2A (0.41) CTSK
SCHEMBL8744699 0.72 CTSS (0.61) CTSKKMO
SCHEMBL9876453 0.72 ALDH1A1 (0.46) C1R
SCHEMBL8744801 0.71 NUDT1 (0.38) AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0653421-B1 Process for preparing 2-cyanoimidazole compounds ISHIHARA SANGYO KAISHA (JP) 1997-01-15 EP disclosed
US-5552557-A Process for preparing 2-cyanoimidazole compounds by reaction of an amino ketone compound ISHIHARA SANGYO KAISHA, LTD. (JP) 1996-09-03 US disclosed
EP-0653421-A1 Process for preparing 2-cyanoimidazole compounds ISHIHARA SANGYO KAISHA LTD. (JP) 1995-05-17 EP disclosed