SCHEMBL8744801

SCHEMBL8744801

Cc1cccc(-c2c[nH]c(C#N)n2)c1C

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 5/20 0.38
USP8 P40818 1/20 0.36
LRRK2 Q5S007 3/20 0.36
TLR8 Q9NR97 1/20 0.34
CNR2 P34972 1/20 0.33
AR P10275 2/20 0.33
NISCH Q9Y2I1 1/20 0.33
ADORA2A P29274 1/20 0.32
TSHR P16473 1/20 0.32
PIK3CD O00329 1/20 0.31
PIK3CA P42336 1/20 0.31
PIK3CB P42338 1/20 0.31
PIK3CG P48736 1/20 0.31
PRKDC P78527 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8744776 0.87 LRRK2 (0.43) USP8LRRK2ARTSHR
SCHEMBL31218523 0.76 TRPA1 (0.40) LRRK2PRKDC
SCHEMBL8744748 0.74 IDO1 (0.41)
SCHEMBL8744696 0.74 L3MBTL1 (0.46) LRRK2ADORA2A
SCHEMBL8744753 0.73 CTSS (0.49) LRRK2ARADORA2ATSHR
SCHEMBL7142089 0.72 TNKS (0.39) NUDT1ARTSHR
SCHEMBL11048748 0.72 NUDT1 (0.38) NUDT1TLR8CNR2ARTSHR
SCHEMBL27857839 0.71 IDO1 (0.41) LRRK2ARNISCH
SCHEMBL8744742 0.70 CYP11B1 (0.43) LRRK2ADORA2A
SCHEMBL25357822 0.70 USP8 (0.38) USP8LRRK2ARTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0653421-B1 Process for preparing 2-cyanoimidazole compounds ISHIHARA SANGYO KAISHA (JP) 1997-01-15 EP disclosed
US-5552557-A Process for preparing 2-cyanoimidazole compounds by reaction of an amino ketone compound ISHIHARA SANGYO KAISHA, LTD. (JP) 1996-09-03 US disclosed
EP-0653421-A1 Process for preparing 2-cyanoimidazole compounds ISHIHARA SANGYO KAISHA LTD. (JP) 1995-05-17 EP disclosed