SCHEMBL8744970

SCHEMBL8744970

O=C(O)Cc1ccc(CN2CCN(c3ccccc3F)CC2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1G O43497 1/20 0.57
ALDH1A1 P00352 5/20 0.57
KDM4E B2RXH2 5/20 0.57
POLB P06746 2/20 0.57
TSHR P16473 1/20 0.57
HSD17B10 Q99714 1/20 0.56
TDP1 Q9NUW8 3/20 0.55
DRD4 P21917 2/20 0.54
DRD3 P35462 2/20 0.54
DRD2 P14416 1/20 0.54
GAA P10253 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
CHRM4 P08173 1/20 0.54
LMNA P02545 1/20 0.53
MAPT P10636 1/20 0.53
KMT2A Q03164 1/20 0.52
ITGB3 P05106 2/20 0.52
ITGA2B P08514 2/20 0.52
ADRA1D P25100 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8745014 0.99 CACNA1G (0.56) CACNA1GALDH1A1KDM4EPOLBTSHR
SCHEMBL13568797 0.85 ALDH1A1 (0.71) ALDH1A1KDM4EPOLBTSHRHSD17B10
SCHEMBL8745020 0.84 ITGB3 (0.52) ALDH1A1TDP1DRD4DRD3DRD2
SCHEMBL8744984 0.84 ATM (0.70) ALDH1A1KDM4EDRD4DRD2SMN1; SMN2
Hydrochloric Acid SCHEMBL8745009 0.83 ATM (0.68) ALDH1A1KDM4EDRD4DRD2SMN1; SMN2
SCHEMBL8691440 0.81 DRD4 (0.70) CACNA1GALDH1A1DRD4DRD3DRD2
SCHEMBL22533031 0.81 KDM4E (0.65) CACNA1GALDH1A1KDM4EPOLBTSHR
SCHEMBL29378232 0.81 KDM4E (0.65) CACNA1GALDH1A1KDM4EPOLBTSHR
SCHEMBL8744973 0.81 MAPK1 (0.70) ALDH1A1KDM4EPOLBTSHRDRD4
Hydrochloric Acid SCHEMBL8690310 0.80 DRD4 (0.68) CACNA1GDRD4DRD3DRD2ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0753515-A2 Benzylpiperazine derivatives as antiallergic and anti-inflammatory agents Senju Pharmaceutical Co., Ltd. (JP) 1997-01-15 EP claimed
EP-0753515-A2 Benzylpiperazine derivatives as antiallergic and anti-inflammatory agents Senju Pharmaceutical Co., Ltd. (JP) 1997-01-15 EP disclosed