SCHEMBL8767407

SCHEMBL8767407

COC(=O)N(Cc1ccccc1)[C@H]1Cc2cc(OC)ccc2C[C@@H]1C

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.41
ACHE P22303 6/20 0.41
GRIN1 Q05586 1/20 0.40
GRIN2B Q13224 1/20 0.40
BCHE P06276 2/20 0.40
MMP1 P03956 3/20 0.40
MMP13 P45452 3/20 0.40
MMP2 P08253 1/20 0.40
MMP3 P08254 1/20 0.40
MMP7 P09237 1/20 0.40
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
MTNR1A P48039 4/20 0.39
MMP9 P14780 2/20 0.39
MTNR1B P49286 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8768044 0.82 METAP1 (0.45) TSHRACHEBCHEMTNR1AMTNR1B
SCHEMBL8768151 0.80 DRD2 (0.52) ACHEGRIN1GRIN2BCA1CA2
SCHEMBL8768766 0.75 ACHE (0.45) TSHRACHEBCHEMTNR1AMTNR1B
SCHEMBL8767508 0.74 ACHE (0.46) TSHRACHEBCHEMTNR1AMTNR1B
SCHEMBL5370790 0.72 KMT2A (0.48) TSHR
SCHEMBL691404 0.69 SLC6A2 (0.52)
SCHEMBL1027731 0.69 DRD2 (0.50) ACHECA1CA2MTNR1AMTNR1B
Hydrochloric Acid SCHEMBL1504396 0.68 SLC6A2 (0.51)
SCHEMBL8768757 0.68 DRD2 (0.42) ACHE
SCHEMBL27596342 0.67 CCR5 (0.48) MMP1MMP13MMP2MMP3MMP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0579833-B1 ETHANOLAMINE DERIVATIVES WITH ANTI-POLLAKIURIA ACTIVITY FUJISAWA PHARMACEUTICAL CO (JP) 1997-08-20 EP disclosed
EP-0579833-A1 ETHANOLAMINE DERIVATIVES WITH ANTI-POLLAKIURIA ACTIVITY. FUJISAWA PHARMACEUTICAL CO (JP) 1994-01-26 EP disclosed
WO-1992018461-A1 ETHANOLAMINE DERIVATIVES WITH ANTI-POLLAKIURIA ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-10-29 WO disclosed