SCHEMBL876986

SCHEMBL876986

CCc1ccc(N(C(CCN2C(=O)c3ccc(C)cc3C2=O)C(=O)O)S(C)(=O)=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.44
CA2 P00918 4/20 0.44
CA9 Q16790 3/20 0.44
CA4 P22748 2/20 0.44
MMP2 P08253 4/20 0.41
MMP9 P14780 4/20 0.41
CA12 O43570 1/20 0.41
MMP3 P08254 1/20 0.40
MMP13 P45452 1/20 0.40
CHRM2 P08172 2/20 0.38
HCRTR2 O43614 1/20 0.37
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37
POLB P06746 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL877006 0.89 MMP2 (0.51) MMP2MMP9MMP3MMP13
SCHEMBL874167 0.88 LPAR1 (0.49) CA1CA2CA9CA4MMP2
SCHEMBL877694 0.87 MMP2 (0.47) CA1CA2CA9CA4MMP2
SCHEMBL874425 0.86 MMP2 (0.48) CA1CA2CA9CA4MMP2
SCHEMBL876861 0.78 MMP2 (0.55) MMP2MMP9MMP3MMP13
SCHEMBL877880 0.77 GPR139 (0.44) NPC1RAB9A
SCHEMBL877277 0.77 MMP2 (0.49) MMP2MMP9MMP3MMP13
SCHEMBL876385 0.75 MMP2 (0.59) MMP2MMP9MMP3MMP13POLB
SCHEMBL877592 0.73 MMP2 (0.41) CA1CA2CA9CA4MMP2
SCHEMBL877131 0.73 MMP2 (0.64) MMP2MMP9MMP3MMP13POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619179-A1 MATRIX METALLOPROTEINASE INHIBITORS Ranbaxy Laboratories Limited (IN) 2013-07-31 EP disclosed
WO-2012038944-A1 MATRIX METALLOPROTEINASE INHIBITORS RANBAXY LABORATORIES LIMITED (IN) 2012-03-29 WO disclosed