SCHEMBL877592

SCHEMBL877592

C=CCOC(=O)C(CCN1C(=O)c2ccc(C)cc2C1=O)N(c1ccc(-c2ccc(Cl)cc2)cc1)S(C)(=O)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 12/20 0.41
MMP9 P14780 12/20 0.41
MMP3 P08254 2/20 0.34
MMP13 P45452 2/20 0.34
MMP1 P03956 1/20 0.34
MMP14 P50281 1/20 0.34
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA9 Q16790 2/20 0.34
CA4 P22748 1/20 0.34
NPSR1 Q6W5P4 2/20 0.33
CA12 O43570 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HTT P42858 1/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL874425 0.86 MMP2 (0.48) MMP2MMP9MMP3MMP13CA1
SCHEMBL876802 0.80 RORC (0.36) MMP2MMP9
SCHEMBL876803 0.80 RORC (0.36) MMP2MMP9
SCHEMBL874167 0.75 LPAR1 (0.49) MMP2MMP9MMP3MMP13CA1
SCHEMBL877694 0.74 MMP2 (0.47) MMP2MMP9MMP3MMP13MMP1
SCHEMBL876986 0.73 CA1 (0.44) MMP2MMP9MMP3MMP13CA1
SCHEMBL876861 0.69 MMP2 (0.55) MMP2MMP9MMP3MMP13MMP1
SCHEMBL873973 0.67 KDM4E (0.42) MMP2MMP9MMP3MMP13MMP1
SCHEMBL877131 0.66 MMP2 (0.64) MMP2MMP9MMP3MMP13MMP1
SCHEMBL877194 0.66 RAB9A (0.35) HTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619179-A1 MATRIX METALLOPROTEINASE INHIBITORS Ranbaxy Laboratories Limited (IN) 2013-07-31 EP disclosed
WO-2012038944-A1 MATRIX METALLOPROTEINASE INHIBITORS RANBAXY LABORATORIES LIMITED (IN) 2012-03-29 WO disclosed