SCHEMBL8774180

SCHEMBL8774180

COc1ccc(CCc2cc(F)c(F)nc2F)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.47
TUBB4A P04350 1/20 0.45
TUBB P07437 1/20 0.45
TUBA3C P0DPH7 1/20 0.45
TUBA1B P68363 1/20 0.45
TUBA4A P68366 1/20 0.45
TUBB4B P68371 1/20 0.45
TUBB3 Q13509 1/20 0.45
TUBB2A Q13885 1/20 0.45
TUBB8 Q3ZCM7 1/20 0.45
TUBA3E Q6PEY2 1/20 0.45
TUBA1A Q71U36 1/20 0.45
TUBA1C Q9BQE3 1/20 0.45
TUBB6 Q9BUF5 1/20 0.45
TUBB2B Q9BVA1 1/20 0.45
TUBB1 Q9H4B7 1/20 0.45
ABCB1 P08183 2/20 0.44
CALM1 P0DP23 2/20 0.44
MAOB P27338 2/20 0.44
PDGFRB P09619 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774796 0.85 NQO1 (0.41) MAOBALDH1A1KDM4EHPGD
SCHEMBL8774833 0.82 LMNA (0.44) RAB9AMAPTL3MBTL1NPC1ALDH1A1
SCHEMBL8775001 0.82 PKM (0.42) ALDH1A1MEN1KMT2A
SCHEMBL8775165 0.82 TAAR1 (0.42) TAAR1RAB9AL3MBTL1NPC1HTT
SCHEMBL8774829 0.82 RAB9A (0.36) RAB9AMAPTNPC1ALDH1A1
SCHEMBL8774157 0.81 RAB9A (0.39) RAB9AMAPTL3MBTL1NPC1ALDH1A1
SCHEMBL9155931 0.79 TAAR1 (0.44) TAAR1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL8774498 0.79 HTR2A (0.40) RAB9ANPC1ALDH1A1KDM4EHPGD
SCHEMBL8774925 0.79 CYP2D6 (0.46) RAB9AMAPTL3MBTL1NPC1ALDH1A1
SCHEMBL8774847 0.79 ACACB (0.43) RAB9AMAPTL3MBTL1NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed