SCHEMBL8774425

SCHEMBL8774425

CCCCCOc1ccc(CCc2cnc(Cl)c(Cl)c2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.46
MAPT P10636 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.44
NPC1 O15118 3/20 0.44
HSD17B10 Q99714 1/20 0.44
GLA P06280 1/20 0.44
MEN1 O00255 1/20 0.44
USP2 O75604 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAPK1 P28482 1/20 0.44
CASP1 P29466 1/20 0.44
KMT2A Q03164 1/20 0.44
SLCO1B3 Q9NPD5 1/20 0.44
SLCO1B1 Q9Y6L6 1/20 0.44
TP53 P04637 1/20 0.43
HPGD P15428 1/20 0.43
NR5A1 Q13285 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774856 0.97 SMN1; SMN2 (0.47) RAB9AMAPTL3MBTL1SMN1; SMN2NPC1
SCHEMBL8774078 0.92 LMNA (0.47) RAB9AMAPTL3MBTL1SMN1; SMN2NPC1
SCHEMBL8774662 0.87 RAB9A (0.46) RAB9AMAPTL3MBTL1SMN1; SMN2NPC1
SCHEMBL8774190 0.85 ALDH1A1 (0.51) RAB9AMAPTL3MBTL1SMN1; SMN2MEN1
SCHEMBL8774663 0.85 SMN1; SMN2 (0.45) RAB9AMAPTL3MBTL1SMN1; SMN2NPC1
SCHEMBL8774683 0.82 RAB9A (0.40) RAB9AMAPTSMN1; SMN2NPC1HSD17B10
SCHEMBL9155401 0.81 RAB9A (0.49) RAB9AMAPTL3MBTL1SMN1; SMN2NPC1
SCHEMBL8774768 0.80 NPC1 (0.54) RAB9AL3MBTL1SMN1; SMN2NPC1HSD17B10
SCHEMBL11667261 0.80 NR5A1 (0.62) RAB9ASMN1; SMN2NPC1MEN1USP2
SCHEMBL8774531 0.79 NPC1 (0.52) RAB9AL3MBTL1SMN1; SMN2NPC1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed