SCHEMBL8774190

SCHEMBL8774190

CCOc1ccc(CCc2cnc(Cl)c(Cl)c2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.51
LMNA P02545 2/20 0.51
POLB P06746 2/20 0.51
MAPT P10636 5/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.46
KDM4E B2RXH2 1/20 0.46
HPGD P15428 1/20 0.46
NQO1 P15559 1/20 0.44
KMT2A Q03164 3/20 0.43
GPR84 Q9NQS5 1/20 0.42
MEN1 O00255 2/20 0.40
PDGFRB P09619 1/20 0.40
PDGFRA P16234 1/20 0.40
THRB P10828 1/20 0.40
SLC5A1 P13866 1/20 0.40
SLC5A2 P31639 1/20 0.40
PLA2G1B P04054 1/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774856 0.88 SMN1; SMN2 (0.47) ALDH1A1LMNAMAPTL3MBTL1RAB9A
SCHEMBL8774078 0.88 LMNA (0.47) ALDH1A1LMNAPOLBMAPTL3MBTL1
SCHEMBL8774425 0.85 RAB9A (0.46) ALDH1A1LMNAMAPTL3MBTL1RAB9A
SCHEMBL8774499 0.83 TAAR1 (0.39) ALDH1A1LMNAMAPTL3MBTL1RAB9A
SCHEMBL8774683 0.83 RAB9A (0.40) ALDH1A1POLBMAPTRAB9ASMN1; SMN2
SCHEMBL8774663 0.81 SMN1; SMN2 (0.45) ALDH1A1LMNAPOLBMAPTL3MBTL1
SCHEMBL8774662 0.79 RAB9A (0.46) ALDH1A1LMNAMAPTL3MBTL1RAB9A
SCHEMBL9154338 0.79 RAB9A (0.50) ALDH1A1LMNAMAPTL3MBTL1RAB9A
SCHEMBL8774722 0.78 ALDH1A1 (0.53) ALDH1A1LMNAPOLBMAPTL3MBTL1
SCHEMBL28616323 0.77 NQO1 (0.74) LMNASMN1; SMN2NQO1GPR84SLC5A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed