SCHEMBL8779100

SCHEMBL8779100

CC(C)C[C@H](N)C(=O)NC(=O)Oc1nccc(OC2CCCCC2)c1O

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LNPEP Q9UIQ6 7/20 0.42
ACACB O00763 2/20 0.40
AAK1 Q2M2I8 7/20 0.38
CIT O14578 3/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779175 0.89 ACACB (0.41) LNPEPACACBPDE4APDE4BPDE4C
SCHEMBL8779229 0.88 IRAK4 (0.40) LNPEPACACBAAK1
SCHEMBL8779239 0.86 LNPEP (0.40) LNPEPAAK1
SCHEMBL8886295 0.84 LNPEP (0.43) LNPEPACACBAAK1CITPDE4A
SCHEMBL8779223 0.81 AAK1 (0.39) AAK1CIT
SCHEMBL8779254 0.81 ACACB (0.38) ACACBPDE4APDE4BPDE4CPDE4D
SCHEMBL8779387 0.79 AAK1 (0.38) AAK1CIT
SCHEMBL8779220 0.79 AAK1 (0.40) LNPEPAAK1CIT
SCHEMBL8779334 0.78 LNPEP (0.42) LNPEPAAK1CIT
SCHEMBL8779428 0.77 IRAK4 (0.43) ACACBPDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed