SCHEMBL8779175

SCHEMBL8779175

C[C@H](N)C(=O)NC(=O)Oc1nccc(OC2CCCCC2)c1O

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACACB O00763 2/20 0.41
LNPEP Q9UIQ6 4/20 0.37
PDE4D Q08499 6/20 0.36
PDE4A P27815 5/20 0.36
PDE4B Q07343 4/20 0.36
PDE4C Q08493 4/20 0.36
CYP19A1 P11511 1/20 0.36
KMO O15229 2/20 0.35
LRRK2 Q5S007 2/20 0.34
IRAK4 Q9NWZ3 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779100 0.89 LNPEP (0.42) ACACBLNPEPPDE4DPDE4APDE4B
SCHEMBL8779428 0.85 IRAK4 (0.43) ACACBPDE4DPDE4APDE4BPDE4C
SCHEMBL8779243 0.84 PPARG (0.38) ACACBLNPEPIRAK4
SCHEMBL8779254 0.83 ACACB (0.38) ACACBPDE4DPDE4APDE4BPDE4C
SCHEMBL8882835 0.83 PDE4D (0.39) ACACBLNPEPPDE4DPDE4APDE4B
SCHEMBL8779264 0.82 AAK1 (0.35)
SCHEMBL8779267 0.81 ALDH1A1 (0.36) KMOIRAK4
SCHEMBL8779308 0.81 ALDH1A1 (0.36) KMOIRAK4
SCHEMBL8779176 0.80 HPGD (0.38) PDE4DPDE4APDE4BPDE4C
SCHEMBL8779212 0.80 HPGD (0.38) PDE4DPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed