SCHEMBL8779334

SCHEMBL8779334

CC(C)C[C@H](N)C(=O)NC(=O)Oc1nccc(OCCOc2ccccc2)c1O

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LNPEP Q9UIQ6 3/20 0.42
ALDH1A1 P00352 2/20 0.39
LARS1 Q9P2J5 2/20 0.38
GRM2 Q14416 2/20 0.37
AAK1 Q2M2I8 5/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
NPSR1 Q6W5P4 1/20 0.36
SCN9A Q15858 1/20 0.36
CIT O14578 1/20 0.35
ANPEP P15144 1/20 0.34
LAP3 P28838 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779092 0.90 ALDH1A1 (0.41) LNPEPALDH1A1GRM2MEN1KMT2A
SCHEMBL8779162 0.90 ALDH1A1 (0.41) LNPEPALDH1A1GRM2MEN1KMT2A
SCHEMBL8779223 0.88 AAK1 (0.39) LARS1AAK1CIT
SCHEMBL8779220 0.86 AAK1 (0.40) LNPEPLARS1AAK1CIT
SCHEMBL8779387 0.82 AAK1 (0.38) LARS1AAK1CIT
SCHEMBL8779239 0.81 LNPEP (0.40) LNPEPAAK1
SCHEMBL8779250 0.81 MEN1 (0.42) ALDH1A1MEN1KMT2A
SCHEMBL8779164 0.80 KDM4E (0.39) ALDH1A1CITANPEP
SCHEMBL8779204 0.80 KDM4E (0.39) ALDH1A1CITANPEP
SCHEMBL8779075 0.80 OPRK1 (0.41) ALDH1A1CIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed