SCHEMBL8779254

SCHEMBL8779254

NCC(=O)NC(=O)Oc1nccc(OC2CCCCC2)c1O

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ACACB O00763 3/20 0.38
LOX P28300 1/20 0.38
LOXL2 Q9Y4K0 1/20 0.38
KMO O15229 3/20 0.36
PDE4D Q08499 4/20 0.34
IRAK4 Q9NWZ3 1/20 0.34
MKNK1 Q9BUB5 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
PDE4A P27815 3/20 0.33
PDE4B Q07343 2/20 0.33
PDE4C Q08493 2/20 0.33
CYP19A1 P11511 1/20 0.33
AR P10275 1/20 0.33
LRRK2 Q5S007 1/20 0.33
IDO1 P14902 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779225 0.86 PARP15 (0.40) ACACBKMOIRAK4
SCHEMBL8786891 0.85 MKNK1 (0.39) ACACBLOXLOXL2PDE4DMKNK1
SCHEMBL8779390 0.84 NFE2L2 (0.38) IDO1
SCHEMBL8779175 0.83 ACACB (0.41) ACACBKMOPDE4DIRAK4PDE4A
SCHEMBL8882242 0.82 LOX (0.39) ACACBLOXLOXL2KMOPDE4D
SCHEMBL8779100 0.81 LNPEP (0.42) ACACBPDE4DPDE4APDE4BPDE4C
SCHEMBL8779326 0.79 SMN1; SMN2 (0.39) ACACB
SCHEMBL8779283 0.77 ALDH1A1 (0.35) IRAK4
SCHEMBL8779273 0.77 IKBKB (0.38) ACACB
SCHEMBL8779237 0.76 LOX (0.36) ACACBLOXLOXL2MKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed