SCHEMBL8779162

SCHEMBL8779162

C[C@H](N)C(=O)NC(=O)Oc1nccc(OCCOc2ccccc2)c1O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
LTA4H P09960 1/20 0.38
LNPEP Q9UIQ6 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
GRM2 Q14416 2/20 0.38
FAAH O00519 1/20 0.36
RAB9A P51151 2/20 0.36
MAPT P10636 1/20 0.36
CARM1 Q86X55 2/20 0.36
PRMT6 Q96LA8 2/20 0.36
XIAP P98170 1/20 0.36
TSHR P16473 2/20 0.36
NPC1 O15118 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PARP10 Q53GL7 1/20 0.35
MAPK1 P28482 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MTNR1A P48039 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779092 1.00 ALDH1A1 (0.41) ALDH1A1MEN1KMT2ALTA4HLNPEP
SCHEMBL8779334 0.90 LNPEP (0.42) ALDH1A1MEN1KMT2ALNPEPNPSR1
SCHEMBL8779136 0.87 IKBKB (0.37) ALDH1A1LTA4HRAB9AMAPTCARM1
SCHEMBL8779325 0.87 IKBKB (0.37) ALDH1A1LTA4HRAB9AMAPTCARM1
SCHEMBL8779198 0.86 LTA4H (0.46) ALDH1A1LTA4HLNPEPRAB9AMAPT
SCHEMBL8779135 0.86 XIAP (0.40) FAAHCARM1PRMT6XIAPNPC1
SCHEMBL8779278 0.86 HTT (0.39) GRM2CARM1PRMT6MAPK1
SCHEMBL8779157 0.86 XIAP (0.40) FAAHCARM1PRMT6XIAPNPC1
SCHEMBL8779165 0.85 XIAP (0.38) MEN1KMT2ALNPEPMAPTCARM1
SCHEMBL8779140 0.85 REN (0.35) LNPEPCARM1PRMT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed