SCHEMBL8779191

SCHEMBL8779191

N[C@@H](CO)C(=O)NC(=O)Oc1nccc(OCC2CCCCC2)c1O

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 2/20 0.38
CDK2 P24941 3/20 0.37
CCNA2 P20248 2/20 0.37
CCNA1 P78396 2/20 0.37
GUCY1B2 O75343 2/20 0.35
GUCY1A2 P33402 2/20 0.35
GUCY1A1 Q02108 2/20 0.35
GUCY1B1 Q02153 2/20 0.35
PARP10 Q53GL7 3/20 0.35
PARP15 Q460N3 2/20 0.35
ACACB O00763 2/20 0.35
XDH P47989 1/20 0.34
MAPK8 P45983 1/20 0.33
CIT O14578 1/20 0.33
GPR88 Q9GZN0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779229 0.89 IRAK4 (0.40) IRAK4CDK2CCNA2CCNA1GUCY1B2
SCHEMBL8779428 0.89 IRAK4 (0.43) IRAK4PARP10PARP15ACACB
SCHEMBL8779259 0.88 IRAK4 (0.37) IRAK4CDK2CCNA2CCNA1ACACB
SCHEMBL8779225 0.83 PARP15 (0.40) IRAK4CDK2CCNA2CCNA1PARP10
SCHEMBL8779239 0.80 LNPEP (0.40)
SCHEMBL8779243 0.79 PPARG (0.38) IRAK4ACACB
SCHEMBL8779418 0.78 PPARG (0.36) IRAK4ACACB
SCHEMBL8779100 0.77 LNPEP (0.42) ACACBCIT
SCHEMBL8779175 0.74 ACACB (0.41) IRAK4ACACB
SCHEMBL8779390 0.73 NFE2L2 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed