SCHEMBL8780815

SCHEMBL8780815

CCCN(CCOc1ccc(N)cc1)CCc1cc(=O)n(C)c(=O)n1C

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.38
PKM P14618 2/20 0.38
ADORA3 P0DMS8 1/20 0.38
ADORA2B P29275 1/20 0.38
ADORA1 P30542 1/20 0.38
KCNH2 Q12809 2/20 0.38
MCHR1 Q99705 1/20 0.38
BCHE P06276 1/20 0.37
ACHE P22303 1/20 0.37
MAPT P10636 1/20 0.36
CHRNA7 P36544 1/20 0.36
KMT2A Q03164 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
ALDH1A1 P00352 2/20 0.35
POLB P06746 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8780776 0.93 MAOA (0.37) ADORA2APKMADORA3ADORA2BADORA1
SCHEMBL8780940 0.92 ADORA2A (0.43) ADORA2APKMADORA3ADORA2BADORA1
SCHEMBL8780789 0.85 ADORA2A (0.41) ADORA2APKMADORA3ADORA2BADORA1
SCHEMBL8780765 0.85 KCNH2 (0.55) PKMKCNH2ALDH1A1HPGD
SCHEMBL8780867 0.85 KCNH2 (0.43) ADORA2APKMADORA3ADORA2BADORA1
SCHEMBL8781017 0.83 NPC1 (0.48) ADORA3KCNH2ACHEALDH1A1
SCHEMBL8780919 0.82 HRH3 (0.41) ADORA2APKMADORA3ADORA2BADORA1
SCHEMBL8780824 0.82 TDP1 (0.39) ADORA2APKMADORA3ADORA2BADORA1
SCHEMBL8780889 0.81 SLC22A2 (0.40) KCNH2MAPT
SCHEMBL8780990 0.81 KCNH2 (0.39) ADORA2APKMADORA3ADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0697407-B1 Pyrimidinedione derivatives and antiarrhythmic compositions containing same MITSUI TOATSU CHEMICALS (JP) 1997-06-25 EP disclosed
EP-0697407-A1 Pyrimidinedione derivatives and antiarrhythmic compositions containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-02-21 EP disclosed