SCHEMBL8780824

SCHEMBL8780824

CC(C)N(CCOc1ccc(N)cc1)CCc1cc(=O)n(C)c(=O)n1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.39
MCHR1 Q99705 2/20 0.38
KCNH2 Q12809 1/20 0.38
PKM P14618 3/20 0.36
PLA2G7 Q13093 1/20 0.36
ALDH1A1 P00352 5/20 0.33
RXFP1 Q9HBX9 2/20 0.33
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
POLB P06746 1/20 0.33
HPGD P15428 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
LTA4H P09960 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8780750 0.93 TDP1 (0.37) TDP1MCHR1KCNH2PKMPLA2G7
SCHEMBL8780751 0.85 PKM (0.51) KCNH2PKMSMN1; SMN2HPGDLTA4H
SCHEMBL8780867 0.85 KCNH2 (0.43) TDP1MCHR1KCNH2PKMADORA3
SCHEMBL8780940 0.83 ADORA2A (0.43) MCHR1KCNH2PKMADORA3ADORA2A
SCHEMBL8780815 0.82 ADORA2A (0.38) MCHR1KCNH2PKMALDH1A1ADORA3
SCHEMBL8780990 0.81 KCNH2 (0.39) MCHR1KCNH2PKMADORA3ADORA2A
SCHEMBL8780857 0.81 ALDH1A1 (0.34) KCNH2PKMPLA2G7ALDH1A1RXFP1
SCHEMBL8780727 0.80 L3MBTL1 (0.44) PKMALDH1A1POLBKDM4EMAPT
SCHEMBL8780907 0.79 PKM (0.52) TDP1KCNH2PKMALDH1A1SMN1; SMN2
SCHEMBL8780789 0.79 ADORA2A (0.41) MCHR1KCNH2PKMADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0697407-B1 Pyrimidinedione derivatives and antiarrhythmic compositions containing same MITSUI TOATSU CHEMICALS (JP) 1997-06-25 EP disclosed
EP-0697407-A1 Pyrimidinedione derivatives and antiarrhythmic compositions containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-02-21 EP disclosed