SCHEMBL9087771

SCHEMBL9087771

CC1(C)C=C(c2cccnc2)c2cc(S(=O)(=O)c3ccccc3)ccc2O1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.42
NAMPT P43490 10/20 0.40
PTGS2 P35354 1/20 0.40
BACE1 P56817 1/20 0.37
KCNH2 Q12809 1/20 0.37
CYP2C9 P11712 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C19 P33261 2/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
PKM P14618 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RXFP1 Q9HBX9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9088314 0.88 RARA (0.39) HTR6NAMPT
SCHEMBL8797664 0.85 HTR6 (0.37) HTR6NAMPTPTGS2BACE1KCNH2
SCHEMBL8793951 0.84 PTGS2 (0.39) NAMPTPTGS2BACE1KCNH2
SCHEMBL9233065 0.83 CYP11B1 (0.44) NAMPTCYP2C9CYP2C19CYP1A2
SCHEMBL9087775 0.80 ALDH1A1 (0.34) HTR6NAMPTPTGS2BACE1CYP2C9
SCHEMBL9084957 0.79 RAB9A (0.46) PTGS2
SCHEMBL8196440 0.75 CYP11B2 (0.46) BACE1KCNH2LMNA
SCHEMBL8796818 0.73 KDM4E (0.33) HTR6NAMPTPTGS2
SCHEMBL8794852 0.72 CYP11B1 (0.43) KCNH2
SCHEMBL8794632 0.72 BACE1 (0.35) BACE1KCNH2CYP2C9CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5493029-A USEFUL IN TREATING ASTHMA AND HYPERTENSION KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1996-02-20 US disclosed
US-5300511-A Spiro-benzopyran derivatives and useful for treating asthma and hypertension KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1994-04-05 US disclosed
EP-0514942-A1 Novel benzopyran derivatives and processes for the preparation thereof KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1992-11-25 EP disclosed