SCHEMBL8798706

SCHEMBL8798706

COc1ccc2c(c1)oc(=O)n2C(C)N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.43
ALDH1A1 P00352 6/20 0.43
HPGD P15428 3/20 0.43
HSD17B10 Q99714 2/20 0.43
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA9 Q16790 2/20 0.43
CA3 P07451 1/20 0.43
AKR1B1 P15121 1/20 0.43
CA4 P22748 1/20 0.43
CA6 P23280 1/20 0.43
CA5A P35218 1/20 0.43
CA7 P43166 1/20 0.43
CA14 Q9ULX7 1/20 0.43
MET P08581 1/20 0.41
KMO O15229 1/20 0.41
NPC1 O15118 3/20 0.41
MAPT P10636 3/20 0.41
RAB9A P51151 3/20 0.41
POLB P06746 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2955732 0.77 KMO (0.51) KDM4EALDH1A1HPGDHSD17B10CA12
SCHEMBL8296662 0.76 L3MBTL1 (0.60) KDM4EALDH1A1HPGDHSD17B10CA12
SCHEMBL29999740 0.75 KDM4E (0.47) KDM4EALDH1A1HPGDHSD17B10CA12
SCHEMBL8798927 0.72 MET (0.57) ALDH1A1HPGDMETKMOMAPT
SCHEMBL14615583 0.72 MAOB (0.39) ALDH1A1HPGDCA12CA1CA9
Hydrochloric Acid SCHEMBL9157992 0.71 MET (0.56) ALDH1A1HPGDMETKMOMAPT
SCHEMBL4413088 0.70 HPGD (0.59) HPGDMETKMOPOLBSMN1; SMN2
SCHEMBL4067603 0.70 KMO (0.46) KDM4EALDH1A1HPGDHSD17B10CA12
SCHEMBL14199043 0.70 POLB (0.52) ALDH1A1HPGDMETKMOMAPT
SCHEMBL30349961 0.69 ALDH1A1 (0.39) KDM4EALDH1A1HPGDHSD17B10CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0506539-B1 Heterocyclic alkylamides, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 1997-05-02 EP disclosed
EP-0506539-A1 Heterocyclic alkylamides, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1992-09-30 EP disclosed