SCHEMBL7526592

SCHEMBL7526592

CC(=O)Oc1c(C(C)(C)C)cc(OC[Si](C)(C)c2ccc(N(C)C)cc2)cc1C(C)(C)C

nearest known ligand 0.32

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
LMNA P02545 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
TSHR P16473 1/20 0.32
CYP2C19 P33261 1/20 0.32
VCAM1 P19320 5/20 0.32
MAPT P10636 3/20 0.31
SQLE Q14534 2/20 0.31
ALDH1A1 P00352 2/20 0.31
HPGD P15428 1/20 0.31
NR1H4 Q96RI1 1/20 0.30
TP53 P04637 1/20 0.30
HDAC1 Q13547 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7523688 0.89 VCAM1 (0.35) MEN1KMT2ALMNAVCAM1MAPT
SCHEMBL7524217 0.87 VCAM1 (0.37) KMT2ATSHRVCAM1MAPTSQLE
SCHEMBL7518758 0.86 VCAM1 (0.47) VCAM1
SCHEMBL7523672 0.86 BACE1 (0.39) CYP3A4VCAM1MAPTSQLE
SCHEMBL7520303 0.85 VCAM1 (0.33) VCAM1MAPTALDH1A1NR1H4
SCHEMBL8839727 0.85 BACE1 (0.38) CYP1A2CYP2C19VCAM1ALDH1A1HPGD
SCHEMBL7513263 0.83 CA2 (0.41) MEN1KMT2ALMNACYP1A2CYP3A4
SCHEMBL7518926 0.83 SLC6A9 (0.33) MEN1KMT2ALMNACYP1A2CYP3A4
SCHEMBL7522609 0.82 CALM1 (0.33) MEN1KMT2AVCAM1MAPTALDH1A1
SCHEMBL8517276 0.79 ADORA3 (0.35) MEN1KMT2ALMNAMAPTSQLE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0900225-B1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS AVENTIS PHARMA INC (US) 2002-01-30 EP disclosed
US-5608095-A Alkyl-4-silyl-phenols and esters thereof as antiatherosclerotic agents HOECHST MARION ROUSSEL, INC. (US) 1997-03-04 US disclosed