SCHEMBL7520303

SCHEMBL7520303

CNc1ccc([Si](C)(C)COc2cc(C(C)(C)C)c(OC(C)=O)c(C(C)(C)C)c2)cc1

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 7/20 0.33
TOP1 P11387 1/20 0.33
NR1H4 Q96RI1 2/20 0.32
ESRRA P11474 1/20 0.31
GAA P10253 2/20 0.30
ALDH1A1 P00352 1/20 0.30
HSP90AA1 P07900 1/20 0.30
MAPT P10636 1/20 0.30
XBP1 P17861 1/20 0.30
ATM Q13315 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
POLB P06746 1/20 0.30
NLRP3 Q96P20 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7523672 0.87 BACE1 (0.39) VCAM1MAPT
SCHEMBL8839727 0.86 BACE1 (0.38) VCAM1ALDH1A1
SCHEMBL7526592 0.85 MEN1 (0.32) VCAM1NR1H4ALDH1A1MAPT
SCHEMBL7516554 0.83 GAA (0.34) VCAM1TOP1NR1H4GAAMAPT
SCHEMBL7517877 0.83 CA2 (0.41) NR1H4GAAALDH1A1MAPTATM
SCHEMBL8517276 0.80 ADORA3 (0.35) NR1H4GAAALDH1A1MAPTATM
SCHEMBL7521161 0.78 ALDH1A1 (0.42) NR1H4ESRRAGAAALDH1A1MAPT
SCHEMBL7522909 0.78 HTT (0.39) TOP1GAAALDH1A1HSP90AA1MAPT
SCHEMBL7524096 0.75 VCAM1 (0.38) VCAM1MAPT
SCHEMBL7523688 0.74 VCAM1 (0.35) VCAM1GAAALDH1A1MAPTXBP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0900225-B1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS AVENTIS PHARMA INC (US) 2002-01-30 EP disclosed
US-5608095-A Alkyl-4-silyl-phenols and esters thereof as antiatherosclerotic agents HOECHST MARION ROUSSEL, INC. (US) 1997-03-04 US disclosed