SCHEMBL8891630

SCHEMBL8891630

CCC(=O)c1c[nH]c2c(-c3ccccc3)cccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
LMNA P02545 2/20 0.52
HTT P42858 1/20 0.52
MAPT P10636 3/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
RAB9A P51151 2/20 0.49
NPC1 O15118 1/20 0.49
MAPK1 P28482 1/20 0.49
CASP3 P42574 1/20 0.49
SENP7 Q9BQF6 1/20 0.49
CNR2 P34972 1/20 0.46
BRPF1 P55201 1/20 0.43
MTNR1A P48039 3/20 0.43
MTNR1B P49286 3/20 0.43
SMN1; SMN2 Q16637 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TUBB4A P04350 2/20 0.41
TUBB P07437 2/20 0.41
TUBA3C P0DPH7 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16453789 0.79 ALDH1A1 (0.80) ALDH1A1LMNAHTTMAPTMEN1
SCHEMBL13715378 0.79 BRPF1 (0.69) ALDH1A1LMNAHTTMAPTMEN1
SCHEMBL8889664 0.79 L3MBTL1 (0.49) ALDH1A1LMNAHTTMAPTMEN1
SCHEMBL27539295 0.78 CNR2 (0.47) ALDH1A1LMNAHTTMAPTMEN1
SCHEMBL8889718 0.78 LMNA (0.56) ALDH1A1LMNAHTTMAPTMEN1
SCHEMBL30505632 0.74 BCAT2 (0.57) ALDH1A1LMNAMAPTMEN1KMT2A
SCHEMBL3420505 0.74 BCAT2 (0.57) ALDH1A1LMNAMAPTMEN1KMT2A
SCHEMBL1903034 0.73 ADAM17 (0.66) ALDH1A1LMNAHTTMAPTMEN1
SCHEMBL27539512 0.73 BCAT2 (0.55) ALDH1A1LMNAMAPTMEN1KMT2A
SCHEMBL28041539 0.72 PARP1 (0.57) ALDH1A1MAPK1CNR2NR4A2FEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997006144-A1 2-CARBOCYCLIC AND 2-HETEROCYCLIC QUINOLINE-4-CARBOXYLIC ACIDS AND SALTS THEREOF USEFUL AS IMMUNOSUPPRESSIVE AGENTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-02-20 WO disclosed
US-5578609-A INHIBITORS OF DIHYDROOROTATE DEHYDROGENASE, ANTITUMOR, TREATMENT OF ORGAN REJECTION THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1996-11-26 US disclosed
US-5523408-A USED FOR TREATMENT OR PREVENTION OF ORGAN TRANSPLANT REJECTION, GRAFT VERSUS HOST DISEASE, CHRONIC INFLAMMATORY DISEASES LIKE PSORIASIS, RHEUMATOID ARTHRITIS IN MAMMAL THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1996-06-04 US disclosed