SCHEMBL8909367

SCHEMBL8909367

NC(=O)C(CN(C(=O)c1cc2ccccc2[nH]1)[C@@H](CC1CCCCC1)[C@@H](O)[C@@H](O)C1CC1)c1cscn1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
P2RX1 P51575 1/20 0.42
F2R P25116 1/20 0.37
REN P00797 2/20 0.35
AKR1C3 P42330 2/20 0.35
MDM2 Q00987 1/20 0.34
KDM4E B2RXH2 2/20 0.34
HSD17B10 Q99714 2/20 0.34
APAF1 O14727 1/20 0.34
TSHR P16473 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
OPRK1 P41145 1/20 0.34
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
CCKBR P32239 1/20 0.32
AR P10275 1/20 0.31
MAOB P27338 1/20 0.31
TP53 P04637 1/20 0.31
NCOA1 Q15788 1/20 0.31
NCOA3 Q9Y6Q9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8910706 0.88 F2R (0.38) P2RX1F2RRENAKR1C3MDM2
SCHEMBL8909363 0.84 P2RX1 (0.52) P2RX1F2RRENAKR1C3MDM2
SCHEMBL8910700 0.76 REN (0.40) P2RX1F2RRENAKR1C3MDM2
SCHEMBL8908848 0.72 F2R (0.37) P2RX1F2RRENAKR1C3MDM2
SCHEMBL8909154 0.68 REN (0.41) P2RX1F2RREN
SCHEMBL8910563 0.67 REN (0.41) P2RX1RENKDM4EHSD17B10TSHR
SCHEMBL8909458 0.67 PYGL (0.36) P2RX1RENAKR1C3KDM4EAR
SCHEMBL8909221 0.66 P2RX1 (0.45) P2RX1REN
SCHEMBL8910552 0.66 REN (0.36) P2RX1F2RREN
SCHEMBL8910252 0.66 KDM4E (0.39) RENAKR1C3KDM4EHSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5688946-A DIPEPTIDES FOR HYPOTENSIVE AGENTS AND CARDIOVASCULAR DISORDERS HOFFMANN LA ROCHE INC. (US) 1997-11-18 US disclosed