SCHEMBL8918109

SCHEMBL8918109

Cn1c(=O)oc2cc(C(=O)CN3CCN(c4ccc(F)cc4)CC3)cnc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
MAPT P10636 3/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C19 P33261 1/20 0.50
SLC6A2 P23975 1/20 0.50
HTR2A P28223 1/20 0.50
SLC6A4 P31645 1/20 0.50
SLC6A3 Q01959 1/20 0.50
GAA P10253 1/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
HTT P42858 2/20 0.45
KDM4E B2RXH2 1/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.43
DEGS1 O15121 1/20 0.43
HTR1A P08908 1/20 0.43
NPC1 O15118 1/20 0.42
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8919693 0.90 POLB (0.46) ALDH1A1MAPTKDM4EHTR1A
SCHEMBL8919198 0.83 POLB (0.47) ALDH1A1MAPTHTR2AGAASMN1; SMN2
SCHEMBL8629045 0.83 ALDH1A1 (0.41) ALDH1A1MAPTHTTMAPK1
SCHEMBL8920278 0.82 MEN1 (0.51) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL8919157 0.80 ALDH1A1 (0.35) ALDH1A1MAPTGAAHTTKDM4E
SCHEMBL8919271 0.80 ALDH1A1 (0.53) ALDH1A1MAPTCYP3A4CYP2D6CYP2C19
SCHEMBL8921274 0.76 ALDH1A1 (0.45) ALDH1A1MAPTCYP3A4CYP2D6CYP2C19
SCHEMBL10392903 0.74 HTR2A (0.64) MAPTSLC6A2HTR2ASLC6A4SLC6A3
SCHEMBL8917897 0.73 SIGMAR1 (0.42) ALDH1A1GAASMN1; SMN2KDM4EMAPK1
SCHEMBL8625701 0.72 ALDH1A1 (0.40) ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5618819-A ANALGESICS ADIR ET COMPAGNIE (FR) 1997-04-08 US disclosed
EP-0691339-A1 Amine derivatives of 1,3-dihydro-2H-pyrrolo(2,3-b)pyridin-2-ones and oxazolo(4,5-b)pyridin-2(3H)-ones, their process of preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-01-10 EP disclosed