SCHEMBL8919271

SCHEMBL8919271

Cn1c(=O)oc2cc(C(=O)CN3CCN(Cc4ccccc4)CC3)cnc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.53
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
MAPT P10636 1/20 0.48
MAPK1 P28482 1/20 0.48
CYP2C19 P33261 1/20 0.48
ACHE P22303 2/20 0.46
APP P05067 1/20 0.46
HIF1A Q16665 1/20 0.44
TSHR P16473 1/20 0.44
PRKAB2 O43741 1/20 0.43
PRKAG1 P54619 1/20 0.43
PRKAA2 P54646 1/20 0.43
PRKAA1 Q13131 1/20 0.43
PRKAG3 Q9UGI9 1/20 0.43
PRKAG2 Q9UGJ0 1/20 0.43
PRKAB1 Q9Y478 1/20 0.43
KMT2A Q03164 1/20 0.42
KDM4E B2RXH2 1/20 0.42
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8919693 0.88 POLB (0.46) ALDH1A1MAPTAPPKMT2AKDM4E
SCHEMBL8920278 0.83 MEN1 (0.51) ALDH1A1CYP3A4CYP2D6MAPK1CYP2C19
SCHEMBL8629045 0.83 ALDH1A1 (0.41) ALDH1A1MAPTMAPK1APPKMT2A
SCHEMBL8919157 0.82 ALDH1A1 (0.35) ALDH1A1MAPTKMT2AKDM4EHPGD
SCHEMBL8921274 0.81 ALDH1A1 (0.45) ALDH1A1CYP3A4CYP2D6MAPTMAPK1
SCHEMBL8918109 0.80 ALDH1A1 (0.50) ALDH1A1CYP3A4CYP2D6MAPTMAPK1
SCHEMBL8919198 0.78 POLB (0.47) ALDH1A1MAPTKDM4ETP53POLB
SCHEMBL8918497 0.77 DRD4 (0.53) ALDH1A1KMT2A
SCHEMBL8917897 0.75 SIGMAR1 (0.42) ALDH1A1MAPK1KDM4EL3MBTL1HPGD
SCHEMBL8919081 0.74 PDE1B (0.41) ALDH1A1TSHRKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5618819-A ANALGESICS ADIR ET COMPAGNIE (FR) 1997-04-08 US disclosed
EP-0691339-A1 Amine derivatives of 1,3-dihydro-2H-pyrrolo(2,3-b)pyridin-2-ones and oxazolo(4,5-b)pyridin-2(3H)-ones, their process of preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-01-10 EP disclosed