SCHEMBL8918622

SCHEMBL8918622

Cn1c(=O)oc2cc(CCN3CCCC3)cnc21

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 7/20 0.41
CYP1A2 P05177 2/20 0.40
CYP2D6 P10635 1/20 0.40
TP53 P04637 1/20 0.39
MAPK1 P28482 1/20 0.39
SLC6A3 Q01959 2/20 0.38
HTR1A P08908 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
CYP3A4 P08684 1/20 0.37
TMEM97 Q5BJF2 1/20 0.36
MAOB P27338 1/20 0.36
MBTD1 Q05BQ5 1/20 0.36
L3MBTL3 Q96JM7 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
SYK P43405 1/20 0.35
USP14 P54578 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8919193 0.91 TMEM97 (0.40) HRH3CYP1A2CYP2D6TP53MAPK1
SCHEMBL8918611 0.90 SIGMAR1 (0.41) SLC6A3HTR1ASLC6A2SLC6A4MAOB
SCHEMBL8918424 0.84 HTR1A (0.51) SLC6A3HTR1ASLC6A2SLC6A4SIGMAR1
SCHEMBL8921432 0.84 HTR1A (0.34) TP53SLC6A3HTR1ASLC6A2SLC6A4
SCHEMBL8917996 0.83 SIGMAR1 (0.44) HTR1ASIGMAR1
SCHEMBL8628216 0.81 PDE10A (0.35) L3MBTL1TDP1SYK
SCHEMBL8919081 0.79 PDE1B (0.41) HTR1A
SCHEMBL8630456 0.78 PDE10A (0.36) HTR1AL3MBTL1
SCHEMBL8917938 0.78 PDE1B (0.43) HRH3SIGMAR1SYK
SCHEMBL8624806 0.77 HSD17B10 (0.35) MAPK1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5618819-A ANALGESICS ADIR ET COMPAGNIE (FR) 1997-04-08 US disclosed
EP-0691339-A1 Amine derivatives of 1,3-dihydro-2H-pyrrolo(2,3-b)pyridin-2-ones and oxazolo(4,5-b)pyridin-2(3H)-ones, their process of preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-01-10 EP disclosed