SCHEMBL8934612

SCHEMBL8934612

Cc1ccn2c(C)c(CCc3ccc(NC4=NC(=O)CN4)cc3)nc2c1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TP53 P04637 5/20 0.36
POLB P06746 2/20 0.36
RXFP1 Q9HBX9 1/20 0.36
THRB P10828 1/20 0.35
MAPT P10636 9/20 0.35
GAA P10253 9/20 0.35
KMT2A Q03164 3/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
HTT P42858 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 1/20 0.34
MITF O75030 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
AOC3 Q16853 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8934556 0.82 ADRA2A (0.48) AOC3
SCHEMBL8934581 0.80 TP53 (0.36) TP53POLBRXFP1THRBMAPT
SCHEMBL8934592 0.74 MAPT (0.37) TP53POLBRXFP1THRBMAPT
SCHEMBL8934533 0.74 NPY1R (0.50) POLBGAASMN1; SMN2ALDH1A1AOC3
Hydrochloric Acid SCHEMBL8934527 0.73 CRHBP (0.40) TP53POLBRXFP1THRBMAPT
SCHEMBL8934510 0.72 NPC1 (0.41) TP53POLBRXFP1THRBMAPT
SCHEMBL8934521 0.72 THRB (0.39) TP53POLBRXFP1THRBMAPT
SCHEMBL9380526 0.69 ALDH1A1 (0.44) TP53POLBRXFP1THRBMAPT
SCHEMBL8934538 0.67 ALDH1A1 (0.48) TP53POLBRXFP1MAPTGAA
SCHEMBL9375701 0.66 DNMT1 (0.35) TP53POLBRXFP1THRBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996030350-A1 AMIDINE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-10-03 WO disclosed