SCHEMBL8942653

SCHEMBL8942653

COc1ccc(C(=O)N(O)CCNC(N)=O)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 5/20 0.47
CA2 P00918 5/20 0.47
PARP10 Q53GL7 2/20 0.47
PARP1 P09874 1/20 0.47
PARP2 Q9UGN5 1/20 0.47
PARP4 Q9UKK3 1/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
KDM4E B2RXH2 1/20 0.46
HPGD P15428 1/20 0.46
PKM P14618 1/20 0.44
MTNR1A P48039 3/20 0.43
MTNR1B P49286 2/20 0.43
DRD2 P14416 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
CYP3A4 P08684 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8942429 0.84 PARP10 (0.45) PARP10PARP1PARP2HPGDMTNR1A
SCHEMBL8942753 0.84 PARP1 (0.52) PARP1NPC1RAB9AHPGDMTNR1A
SCHEMBL8942432 0.84 RAB9A (0.46) NPC1RAB9AKMT2A
SCHEMBL8942484 0.83 PARP10 (0.50) CA1CA2PARP10NPC1RAB9A
SCHEMBL8942633 0.81 TP53 (0.52) NPC1RAB9A
SCHEMBL8783847 0.80 NPC1 (0.61) CA1CA2NPC1RAB9AHPGD
SCHEMBL8942623 0.78 HPGD (0.46) NPC1RAB9AKDM4EHPGDDRD2
SCHEMBL8942585 0.74 MEN1 (0.42) PARP10PARP1NPC1RAB9AKDM4E
SCHEMBL31483087 0.72 MTNR1A (0.73) NPC1RAB9AMTNR1AMTNR1BDRD2
SCHEMBL7924560 0.72 SMN1; SMN2 (0.73) NPC1RAB9AKDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5514702-A Arylamidoalkyl-N-hydroxyurea compounds having lipoxygenase inhibitory activity ABBOTT LABORATORIES (US) 1996-05-07 US disclosed