SCHEMBL8942753

SCHEMBL8942753

COc1cccc(C(=O)N(O)CCNC(N)=O)c1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.52
MTNR1A P48039 8/20 0.48
MTNR1B P49286 7/20 0.48
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
GAA P10253 2/20 0.46
HPGD P15428 1/20 0.46
SIGMAR1 Q99720 1/20 0.46
PRSS1 P07477 1/20 0.46
PRSS2 P07478 1/20 0.46
PRSS3 P35030 1/20 0.46
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
MMP13 P45452 1/20 0.44
TDP1 Q9NUW8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8942429 0.92 PARP10 (0.45) PARP1MTNR1AMTNR1BMEN1KMT2A
SCHEMBL8942585 0.88 MEN1 (0.42) PARP1MEN1KMT2AGAAPRSS1
SCHEMBL8942653 0.84 CA1 (0.47) PARP1MTNR1AMTNR1BCES2CES1
SCHEMBL8942260 0.83 FURIN (0.39) MTNR1AMTNR1BKMT2AALDH1A1
SCHEMBL8942395 0.83 ALOX5 (0.47) ALDH1A1
SCHEMBL8942408 0.82 TNKS (0.39) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL8942712 0.82 PARP14 (0.45) MEN1KMT2A
SCHEMBL8783271 0.82 SIGMAR1 (0.57) PARP1MEN1KMT2AGAAHPGD
SCHEMBL8942679 0.82 MAPT (0.47) MEN1KMT2AHPGDNPC1RAB9A
SCHEMBL8942661 0.81 KMO (0.53) MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5514702-A Arylamidoalkyl-N-hydroxyurea compounds having lipoxygenase inhibitory activity ABBOTT LABORATORIES (US) 1996-05-07 US disclosed