SCHEMBL8963516

SCHEMBL8963516

Cc1ccc(-c2nc(C(C(c3ccc(Cl)cc3)c3ccc(Cl)cc3)N3CCNCC3)c(C)[nH]2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP19A1 P11511 1/20 0.42
OPRM1 P35372 2/20 0.36
OPRD1 P41143 2/20 0.36
CTSS P25774 2/20 0.35
MAPK1 P28482 1/20 0.34
NPY5R Q15761 1/20 0.33
MGAM O43451 1/20 0.33
GAA P10253 1/20 0.33
SI P14410 1/20 0.33
MGAM2 Q2M2H8 1/20 0.33
HTR1A P08908 3/20 0.32
HTR2B P41595 3/20 0.32
HTR7 P34969 2/20 0.32
HTR5A P47898 2/20 0.32
HTR6 P50406 2/20 0.32
HTR3A P46098 2/20 0.32
HTR2A P28223 2/20 0.32
HTR1D P28221 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8964088 0.94 OPRD1 (0.37) CHEK2CYP2D6CYP19A1OPRM1OPRD1
SCHEMBL8963650 0.91 CHEK2 (0.40) CHEK2CYP2D6CYP19A1OPRD1NPY5R
SCHEMBL8963979 0.91 CYP2D6 (0.42) CHEK2CYP2D6CYP19A1OPRM1OPRD1
SCHEMBL8963637 0.89 MAPK13 (0.37) CHEK2CYP2D6OPRM1OPRD1MGAM
SCHEMBL8963580 0.89 PRMT5 (0.40) OPRD1PRMT5
Hydrochloric Acid SCHEMBL8963783 0.88 PRMT5 (0.40) OPRD1PRMT5
SCHEMBL8964138 0.88 SLC6A4 (0.38) CHEK2CYP2D6OPRM1OPRD1CTSS
SCHEMBL8963820 0.87 HDAC6 (0.34) CHEK2OPRM1OPRD1
SCHEMBL8963737 0.87 OPRM1 (0.38) OPRM1OPRD1GAAHTR1AHTR2B
SCHEMBL8963675 0.84 TACR1 (0.36) CHEK2OPRM1OPRD1HTR1AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5514800-A CALCIUM CHANNEL BLOCKERS, CEREBRAL ISCHEMIA SYNTEX PHARMACEUTICALS, LTD. (GB) 1996-05-07 US disclosed