SCHEMBL8964138

SCHEMBL8964138

Cc1ccc(-c2nc(C(C(c3cccc(Cl)c3)c3cccc(Cl)c3)N3CCNCC3)c(C)[nH]2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 9/20 0.38
SLC6A2 P23975 7/20 0.38
CHEK2 O96017 1/20 0.36
TACR1 P25103 2/20 0.35
PIN1 Q13526 1/20 0.35
CTSS P25774 1/20 0.35
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
OPRL1 P41146 1/20 0.34
NPY5R Q15761 1/20 0.34
SLC6A3 Q01959 5/20 0.33
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
ADRB1 P08588 1/20 0.33
CYP3A4 P08684 1/20 0.33
HTR1A P08908 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8963675 0.91 TACR1 (0.36) CHEK2TACR1PIN1OPRM1OPRD1
SCHEMBL8963516 0.88 CHEK2 (0.42) CHEK2CTSSOPRM1OPRD1NPY5R
SCHEMBL8963580 0.87 PRMT5 (0.40) SLC6A4SLC6A2TACR1OPRD1CYP1A2
SCHEMBL8963787 0.87 PIN1 (0.45) SLC6A4SLC6A2TACR1PIN1NPY5R
Hydrochloric Acid SCHEMBL8963783 0.86 PRMT5 (0.40) SLC6A4SLC6A2TACR1OPRD1CYP1A2
SCHEMBL8963532 0.86 SLC6A2 (0.41) SLC6A4SLC6A2TACR1PIN1OPRM1
SCHEMBL8963691 0.86 TACR1 (0.34) SLC6A4CHEK2TACR1OPRD1PRMT5
SCHEMBL8964088 0.86 OPRD1 (0.37) CHEK2OPRM1OPRD1ADRB1HTR1A
SCHEMBL8963650 0.85 CHEK2 (0.40) SLC6A4SLC6A2CHEK2OPRD1NPY5R
SCHEMBL8963679 0.82 MEN1 (0.42) SLC6A4SLC6A2PIN1OPRD1NPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5514800-A CALCIUM CHANNEL BLOCKERS, CEREBRAL ISCHEMIA SYNTEX PHARMACEUTICALS, LTD. (GB) 1996-05-07 US disclosed