SCHEMBL8963532

SCHEMBL8963532

COc1cccc(C(c2cccc(OC)c2)C(c2nc(-c3ccc(C)cc3)[nH]c2C)N2CCNCC2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 3/20 0.41
SLC6A4 P31645 1/20 0.41
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
ADRB1 P08588 1/20 0.38
TACR1 P25103 1/20 0.38
PIN1 Q13526 1/20 0.37
ROCK2 O75116 2/20 0.36
ROCK1 Q13464 2/20 0.36
PRMT5 O14744 1/20 0.36
HTR1A P08908 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR7 P34969 1/20 0.35
HTR2B P41595 1/20 0.35
HTR3A P46098 1/20 0.35
HTR6 P50406 1/20 0.35
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
TP53 P04637 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8963675 0.89 TACR1 (0.36) OPRM1OPRD1ADRB1TACR1PIN1
SCHEMBL8963737 0.88 OPRM1 (0.38) OPRM1OPRD1ADRB1TACR1PRMT5
SCHEMBL8963561 0.87 SLC6A2 (0.47) SLC6A2SLC6A4OPRM1OPRD1ADRB1
SCHEMBL8964138 0.86 SLC6A4 (0.38) SLC6A2SLC6A4OPRM1OPRD1ADRB1
SCHEMBL8964068 0.86 PRMT5 (0.44) SLC6A2SLC6A4OPRM1OPRD1PRMT5
SCHEMBL8963580 0.86 PRMT5 (0.40) SLC6A2SLC6A4OPRD1TACR1PRMT5
Hydrochloric Acid SCHEMBL8963783 0.85 PRMT5 (0.40) SLC6A2SLC6A4OPRD1TACR1PRMT5
SCHEMBL8963691 0.85 TACR1 (0.34) SLC6A4OPRD1TACR1PRMT5
SCHEMBL8964088 0.84 OPRD1 (0.37) OPRM1OPRD1ADRB1PRMT5HTR1A
SCHEMBL8963505 0.81 SLC6A2 (0.41) SLC6A2SLC6A4ADRB1TACR1PRMT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5514800-A CALCIUM CHANNEL BLOCKERS, CEREBRAL ISCHEMIA SYNTEX PHARMACEUTICALS, LTD. (GB) 1996-05-07 US disclosed