SCHEMBL8967876

SCHEMBL8967876

O=CN(CC12CCCN1CCC2)c1ccccc1-c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.37
OPRM1 P35372 6/20 0.35
KCNH2 Q12809 2/20 0.34
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
RAB9A P51151 1/20 0.32
TSHR P16473 1/20 0.31
RECQL P46063 1/20 0.31
ALKBH5 Q6P6C2 2/20 0.31
FTO Q9C0B1 2/20 0.31
OPRK1 P41145 1/20 0.30
ESR1 P03372 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8967955 0.81 SIGMAR1 (0.47) SIGMAR1OPRM1KCNH2RAB9ASLC6A2
SCHEMBL8967541 0.80 SIGMAR1 (0.37) SIGMAR1OPRM1KCNH2ALDH1A1MAPT
SCHEMBL8968097 0.80 SIGMAR1 (0.35) SIGMAR1OPRM1KCNH2ALDH1A1MAPT
SCHEMBL8967658 0.79 SIGMAR1 (0.41) SIGMAR1OPRM1KCNH2ALDH1A1RAB9A
SCHEMBL8967505 0.76 SIGMAR1 (0.35) SIGMAR1OPRM1KCNH2ALDH1A1TSHR
SCHEMBL8967761 0.73 SIGMAR1 (0.40) SIGMAR1OPRM1KCNH2RAB9AALKBH5
SCHEMBL8968027 0.72 TUBB3 (0.36) SIGMAR1ALDH1A1MAPTSMN1; SMN2TSHR
SCHEMBL8967593 0.70 ALDH1A1 (0.33) SIGMAR1OPRM1KCNH2ALDH1A1MAPT
SCHEMBL14471536 0.63 ALDH1A1 (0.38) ALDH1A1SMN1; SMN2SLC6A2SLC6A4SLC6A3
SCHEMBL8967652 0.63 SIGMAR1 (0.41) SIGMAR1OPRM1KCNH2ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5530138-A A PYRROLIZINE DERIVATIVE; EFFECTIVE IN THE TREATMENT OF SENILE DEMENTIA SANWA KAGAKU KENKYUSHO CO., LTD. (JP) 1996-06-25 US claimed
EP-0647642-A1 1-Azabicyclo(3.3.0)octane derivatives and their use SANWA KAGAKU KENKYUSHO CO., LTD. (JP) 1995-04-12 EP claimed
US-5530138-A A PYRROLIZINE DERIVATIVE; EFFECTIVE IN THE TREATMENT OF SENILE DEMENTIA SANWA KAGAKU KENKYUSHO CO., LTD. (JP) 1996-06-25 US disclosed
EP-0647642-A1 1-Azabicyclo(3.3.0)octane derivatives and their use SANWA KAGAKU KENKYUSHO CO., LTD. (JP) 1995-04-12 EP disclosed