SCHEMBL8967955

SCHEMBL8967955

O=CN(CC12CCCN1CCC2)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 13/20 0.47
OPRM1 P35372 11/20 0.44
KCNH2 Q12809 6/20 0.37
RAB9A P51151 1/20 0.35
KDM4E B2RXH2 1/20 0.35
CHRNA7 P36544 1/20 0.33
HCN1 O60741 1/20 0.33
HCN4 Q9Y3Q4 1/20 0.33
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
CYP2B6 P20813 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
PRCP P42785 1/20 0.33
SLC6A3 Q01959 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
GRIN2B Q13224 1/20 0.33
GRIN2C Q14957 1/20 0.33
GRIN3A Q8TCU5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8967658 0.88 SIGMAR1 (0.41) SIGMAR1OPRM1KCNH2RAB9AKDM4E
SCHEMBL8967761 0.85 SIGMAR1 (0.40) SIGMAR1OPRM1KCNH2RAB9AKDM4E
SCHEMBL18458654 0.79 OPRM1 (0.50) SIGMAR1OPRM1KCNH2SLC6A3
SCHEMBL8968097 0.78 SIGMAR1 (0.35) SIGMAR1OPRM1KCNH2KDM4ESLC6A2
SCHEMBL8967505 0.77 SIGMAR1 (0.35) SIGMAR1OPRM1KCNH2CHRNA7SLC6A4
SCHEMBL8967663 0.76 SIGMAR1 (0.47) SIGMAR1OPRM1KCNH2RAB9AKDM4E
SCHEMBL8968027 0.73 TUBB3 (0.36) SIGMAR1KDM4EHCN1HCN4
SCHEMBL21337552 0.72 SIGMAR1 (0.45) SIGMAR1OPRM1KCNH2KDM4EPRCP
SCHEMBL8967652 0.69 SIGMAR1 (0.41) SIGMAR1OPRM1KCNH2KDM4E
SCHEMBL8967593 0.68 ALDH1A1 (0.33) SIGMAR1OPRM1KCNH2KDM4ESLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5530138-A A PYRROLIZINE DERIVATIVE; EFFECTIVE IN THE TREATMENT OF SENILE DEMENTIA SANWA KAGAKU KENKYUSHO CO., LTD. (JP) 1996-06-25 US claimed
EP-0647642-A1 1-Azabicyclo(3.3.0)octane derivatives and their use SANWA KAGAKU KENKYUSHO CO., LTD. (JP) 1995-04-12 EP claimed
US-5530138-A A PYRROLIZINE DERIVATIVE; EFFECTIVE IN THE TREATMENT OF SENILE DEMENTIA SANWA KAGAKU KENKYUSHO CO., LTD. (JP) 1996-06-25 US disclosed
EP-0647642-A1 1-Azabicyclo(3.3.0)octane derivatives and their use SANWA KAGAKU KENKYUSHO CO., LTD. (JP) 1995-04-12 EP disclosed