SCHEMBL8993373

SCHEMBL8993373

Cc1ccccc1Cc1ccc(CC#N)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.43
KMT2A Q03164 3/20 0.40
TAAR1 Q96RJ0 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
MEN1 O00255 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
TSHR P16473 1/20 0.38
ABCB1 P08183 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
KEAP1 Q14145 1/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8095627 0.83 LTA4H (0.53) LTA4HTAAR1SLC6A2SLC6A4SLC6A3
SCHEMBL31426960 0.81 ALDH1A1 (0.47) KMT2ATAAR1MEN1SMN1; SMN2CYP1A2
SCHEMBL102904 0.81 ALDH1A1 (0.47) KMT2ATAAR1MEN1SMN1; SMN2CYP1A2
Water SCHEMBL28641184 0.81 ALDH1A1 (0.47) KMT2ATAAR1MEN1SMN1; SMN2CYP1A2
SCHEMBL27287538 0.79 HTR2A (0.44) KMT2ASLC6A2SLC6A4SLC6A3SMN1; SMN2
SCHEMBL4003141 0.79 KEAP1 (0.63) KMT2ATAAR1MEN1CYP3A4CYP2D6
SCHEMBL8992952 0.79 NPC1 (0.50) LTA4HTAAR1TSHRALDH1A1MAPT
SCHEMBL8993391 0.78 CNR2 (0.44) KMT2AMEN1TSHRLMNAMAPT
SCHEMBL6378299 0.77 POLB (0.51) LTA4HKMT2ATAAR1MEN1CYP3A4
SCHEMBL2140995 0.77 CALM1 (0.57) LTA4HKMT2ATAAR1MEN1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed