SCHEMBL902860

SCHEMBL902860

Nc1cccc(-c2ccccc2CCNC(=O)O)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.43
ASIC3 Q9UHC3 1/20 0.41
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
ATR Q13535 1/20 0.36
NOS3 P29474 4/20 0.36
NOS1 P29475 4/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
MTNR1B P49286 1/20 0.36
F2 P00734 1/20 0.35
PRSS1 P07477 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL902861 0.77 NOS1 (0.53) ASIC3KDM4ELMNAALDH1A1NOS3
SCHEMBL27508570 0.75 ASIC3 (0.46) ASIC3NOS3NOS1
SCHEMBL901874 0.75 ASIC3 (0.47) ASIC3KDM4ELMNANOS3NOS1
SCHEMBL4598193 0.73 MTNR1A (0.46) MTNR1AKDM4EALDH1A1HPGDMTNR1B
SCHEMBL1567114 0.70 MTNR1A (0.73) MTNR1AMTNR1B
SCHEMBL6921461 0.70 CYP1A2 (0.49) MTNR1AKDM4ELMNAMTNR1B
SCHEMBL20773417 0.69 KCNH2 (0.53) ALDH1A1HDAC3HDAC1HDAC2HDAC6
SCHEMBL5309632 0.68 MPO (0.56) KDM4E
SCHEMBL10348018 0.68 ALDH1A1 (0.54) MTNR1ALMNAALDH1A1HPGDMTNR1B
SCHEMBL19212244 0.68 PTGDR2 (0.47) MTNR1AHPGDMTNR1BHDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041476-A1 PYRIDINE AND ISOQUINOLINE DERIVATIVES AS SYK- AND JAK-KINASE INHIBITORS ALMIRALL, S.A. (ES) 2012-04-05 WO disclosed