SCHEMBL902861

SCHEMBL902861

Nc1cccc(-c2ccc(CCNC(=O)O)cc2)n1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 6/20 0.53
NOS3 P29474 5/20 0.53
CHRM2 P08172 1/20 0.52
CHRM4 P08173 1/20 0.52
ASIC3 Q9UHC3 1/20 0.50
HIF1A Q16665 2/20 0.43
MAPT P10636 2/20 0.43
TP53 P04637 1/20 0.43
CA2 P00918 2/20 0.42
CA4 P22748 1/20 0.42
CA9 Q16790 1/20 0.42
SCN2A Q99250 1/20 0.41
SCN10A Q9Y5Y9 1/20 0.41
BRS3 P32247 1/20 0.41
ALDH1A1 P00352 2/20 0.41
THRB P10828 1/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
CA1 P00915 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL901874 0.86 ASIC3 (0.47) NOS1NOS3CHRM2CHRM4ASIC3
SCHEMBL6618736 0.81 NOS1 (0.64) NOS1NOS3CHRM2CHRM4ASIC3
SCHEMBL4582523 0.78 ALDH1A1 (0.56) MAPTALDH1A1KDM4ELMNA
SCHEMBL6622090 0.78 NOS1 (0.60) NOS1NOS3CHRM2CHRM4ASIC3
SCHEMBL5338527 0.77 OPRM1 (0.54)
SCHEMBL23828889 0.77 HCAR2 (0.55) HIF1AMAPTTP53ALDH1A1KDM4E
SCHEMBL902860 0.77 MTNR1A (0.43) NOS1NOS3CHRM2CHRM4ASIC3
SCHEMBL6623818 0.76 NOS1 (0.66) NOS1NOS3CHRM2CHRM4
SCHEMBL6620843 0.76 SIGMAR1 (0.58) NOS1NOS3ASIC3
SCHEMBL6620927 0.76 NOS1 (0.60) NOS1NOS3CHRM2CHRM4ASIC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041476-A1 PYRIDINE AND ISOQUINOLINE DERIVATIVES AS SYK- AND JAK-KINASE INHIBITORS ALMIRALL, S.A. (ES) 2012-04-05 WO disclosed