SCHEMBL9044667

SCHEMBL9044667

O=C(O)CC[C@H](NC(=O)c1ccc(CCn2cnc3nccc-3c2O)cc1)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ATIC P31939 4/20 0.49
SHMT1 P34896 3/20 0.49
SHMT2 P34897 3/20 0.49
DHFR P00374 5/20 0.48
GART P22102 6/20 0.48
CA2 P00918 2/20 0.45
CA1 P00915 1/20 0.45
TYMS P04818 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9047109 0.92 CA2 (0.47) ATICSHMT1SHMT2DHFRGART
SCHEMBL573199 0.86 DHFR (0.52) ATICSHMT1SHMT2DHFRGART
SCHEMBL9045940 0.86 ATIC (0.47) ATICSHMT1SHMT2DHFRGART
SCHEMBL9046201 0.83 TAS1R3 (0.41) ATICSHMT1SHMT2CA2CA1
SCHEMBL9043718 0.81 ATIC (0.43) ATICSHMT1SHMT2DHFRGART
SCHEMBL9044214 0.80 DHFR (0.46) ATICSHMT1SHMT2DHFRGART
SCHEMBL9049515 0.79 CA2 (0.44) ATICSHMT1SHMT2DHFRGART
SCHEMBL9049344 0.79 CA2 (0.43) ATICSHMT1SHMT2DHFRGART
SCHEMBL9046824 0.75 ATIC (0.55) ATICSHMT1SHMT2DHFRGART
SCHEMBL9045484 0.74 CYP4A11 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0432677-B1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives UNIV PRINCETON (US) 1996-03-06 EP claimed
US-4996206-A Antitumor agent THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-02-26 US claimed
JP-8003166-A None JP disclosed
EP-0432677-B1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives UNIV PRINCETON (US) 1996-03-06 EP disclosed
JP-H083166-A N-(PYRROLO(2,3-D)PYRIMIDIN-3-YLACYL)GLUTAMIC ACID DERIVATIVE UNIV PRINCETON 1996-01-09 JP disclosed
US-5426187-A Process for the preparation of 4-hydroxy-5-substituted ethynylpyrrolo [2,3-d]pyrimidine intermediates ELI LILLY AND COMPANY (US) 1995-06-20 US disclosed
US-5344932-A N-(pyrrolo(2,3-d)pyrimidin-3-ylacyl)-glutamic acid derivatives TRUSTEES OF PRINCETON UNIVERSITY (US) 1994-09-06 US disclosed
US-5248775-A Pyrrolo(2,3-d)pyrimidines THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1993-09-28 US disclosed
EP-0432677-A1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-06-19 EP disclosed
US-4996206-A Antitumor agent THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-02-26 US disclosed
US-4996206-A Antitumor agent THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-02-26 US disclosed