SCHEMBL9045940

SCHEMBL9045940

Cc1cc2c(O)n(CCc3ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc3)cnc-2n1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ATIC P31939 4/20 0.47
SHMT1 P34896 3/20 0.47
SHMT2 P34897 3/20 0.47
DHFR P00374 7/20 0.47
GART P22102 6/20 0.47
TYMS P04818 3/20 0.47
FOLR2 P14207 2/20 0.44
FOLR1 P15328 2/20 0.44
SLC46A1 Q96NT5 2/20 0.44
SLC19A1 P41440 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9049515 0.93 CA2 (0.44) ATICSHMT1SHMT2DHFRGART
SCHEMBL573199 0.89 DHFR (0.52) ATICSHMT1SHMT2DHFRGART
SCHEMBL9044667 0.86 ATIC (0.49) ATICSHMT1SHMT2DHFRGART
SCHEMBL9043718 0.86 ATIC (0.43) ATICSHMT1SHMT2DHFRGART
SCHEMBL9471199 0.85 TAS1R3 (0.41)
SCHEMBL9044214 0.83 DHFR (0.46) ATICSHMT1SHMT2DHFRGART
SCHEMBL9047109 0.79 CA2 (0.47) ATICSHMT1SHMT2DHFRGART
SCHEMBL9046824 0.78 ATIC (0.55) ATICSHMT1SHMT2DHFRGART
SCHEMBL9342476 0.78 ATIC (0.48) ATICSHMT1SHMT2DHFRGART
SCHEMBL9045385 0.77 FOLR2 (0.51) ATICSHMT1SHMT2DHFRGART

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0432677-B1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives UNIV PRINCETON (US) 1996-03-06 EP claimed
EP-0432677-A1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-06-19 EP claimed
US-4996206-A Antitumor agent THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-02-26 US claimed
EP-0432677-B1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives UNIV PRINCETON (US) 1996-03-06 EP disclosed
US-5344932-A N-(pyrrolo(2,3-d)pyrimidin-3-ylacyl)-glutamic acid derivatives TRUSTEES OF PRINCETON UNIVERSITY (US) 1994-09-06 US disclosed
US-5248775-A Pyrrolo(2,3-d)pyrimidines THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1993-09-28 US disclosed
EP-0432677-A1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-06-19 EP disclosed
US-4996206-A Antitumor agent THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-02-26 US disclosed