SCHEMBL9045394

SCHEMBL9045394

C[CH]CCCc1c(Cl)cccc1C(C)=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.39
CYP3A4 P08684 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
LIPG Q9Y5X9 1/20 0.36
KMT2A Q03164 2/20 0.36
TSHR P16473 1/20 0.35
HPGD P15428 2/20 0.35
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HTT P42858 1/20 0.34
CD38 P28907 1/20 0.34
TAAR1 Q96RJ0 1/20 0.33
JAK2 O60674 1/20 0.33
ERBB2 P04626 1/20 0.33
MARK3 P27448 1/20 0.33
IRAK1 P51617 1/20 0.33
NEK4 P51957 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9047365 0.88 TSHR (0.46) AKR1B1CYP3A4CYP1A2CYP2C9CYP2C19
SCHEMBL9048247 0.84 GPR52 (0.40) HPGDSMN1; SMN2
SCHEMBL9045397 0.82 GABRA1 (0.35) TSHRHTT
SCHEMBL9045101 0.82 KMT2A (0.39) KMT2ACES2CES1SMN1; SMN2CD38
SCHEMBL9047503 0.81 AKR1B1 (0.41) AKR1B1CYP3A4CYP1A2CYP2C9CYP2C19
SCHEMBL9047469 0.81 CA2 (0.34) TSHRSMN1; SMN2
SCHEMBL9057953 0.79 GABRA1 (0.41) CYP3A4CYP1A2TSHRHPGDSMN1; SMN2
SCHEMBL9046887 0.77 TAAR1 (0.39) AKR1B1LIPGSMN1; SMN2HTTTAAR1
SCHEMBL9046020 0.76 TAAR1 (0.36) AKR1B1LIPGSMN1; SMN2TAAR1
SCHEMBL9045669 0.74 TAAR1 (0.58) KMT2ATSHRSMN1; SMN2HTTTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0690854-A1 1-PHENYL-IMIDAZOL-2-ONE BIPHENYLMETHYL COMPOUNDS FOR TREATMENT OF CIRCULATORY DISORDERS G.D. SEARLE & CO. (US) 1996-01-10 EP disclosed