SCHEMBL9050448

SCHEMBL9050448

O=C(Nc1cnc2ccccc2c1)C1CCc2[nH]cnc2C1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 4/20 0.47
RAB9A P51151 8/20 0.47
MAPT P10636 2/20 0.47
EPHX2 P34913 1/20 0.46
KDR P35968 2/20 0.46
KDM4E B2RXH2 5/20 0.45
NPC1 O15118 7/20 0.44
SMN1; SMN2 Q16637 5/20 0.44
HSD17B10 Q99714 3/20 0.44
TP53 P04637 1/20 0.44
JAK2 O60674 1/20 0.43
CNR2 P34972 1/20 0.43
POLB P06746 2/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.42
TSHR P16473 1/20 0.42
MITF O75030 1/20 0.42
XBP1 P17861 1/20 0.42
PAX8 Q06710 1/20 0.42
KLF5 Q13887 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6851321 0.83 HPGD (0.48) RAB9AMAPTKDM4ENPC1SMN1; SMN2
SCHEMBL6850904 0.82 KDM2B (0.47) CNR2
Fumaric Acid SCHEMBL7334141 0.78 HPGD (0.43) RAB9AMAPTKDM4ENPC1SMN1; SMN2
SCHEMBL9048814 0.78 GSK3A (0.47) RAB9AKDM4ENPC1POLBALDH1A1
SCHEMBL9049386 0.78 CYP1A2 (0.49) RAB9AMAPTKDM4ENPC1SMN1; SMN2
SCHEMBL9050232 0.78 SMN1; SMN2 (0.63) RAB9AMAPTNPC1SMN1; SMN2POLB
Hydrochloric Acid SCHEMBL9051872 0.78 GSK3A (0.46) RAB9AKDM4ENPC1POLBALDH1A1
SCHEMBL9050851 0.76 POLB (0.54) TRPV1RAB9AMAPTKDM4ENPC1
SCHEMBL7327986 0.75 L3MBTL1 (0.47) RAB9AEPHX2KDM4ENPC1SMN1; SMN2
SCHEMBL7325548 0.75 SMN1; SMN2 (0.45) RAB9ANPC1SMN1; SMN2TP53POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0381422-B1 Tetrahydrobenzimidazole derivatives YAMANOUCHI PHARMA CO LTD (JP) 1996-10-23 EP disclosed
US-5496942-A 5-HT3-RECEPTOR ANTAGONISTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-03-05 US disclosed
US-5344927-A 5-HT3 antagonist YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1994-09-06 US disclosed
EP-0381422-A1 Tetrahydrobenzimidazole derivatives YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1990-08-08 EP disclosed