SCHEMBL9050232

SCHEMBL9050232

O=C(Nc1nc2ccccc2[nH]1)C1CCc2[nH]cnc2C1

nearest known ligand 0.63

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 7/20 0.63
NPC1 O15118 7/20 0.61
RAB9A P51151 7/20 0.61
POLB P06746 2/20 0.61
TDP1 Q9NUW8 1/20 0.61
CYP1A2 P05177 1/20 0.51
ADORA2A P29274 2/20 0.51
ADORA1 P30542 1/20 0.51
LPAR2 Q9HBW0 2/20 0.47
LMNA P02545 2/20 0.47
HTT P42858 1/20 0.47
CYP3A4 P08684 1/20 0.46
GSK3A P49840 1/20 0.46
GSK3B P49841 1/20 0.46
PKM P14618 1/20 0.44
MAOB P27338 1/20 0.44
USP2 O75604 1/20 0.44
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6851321 0.79 HPGD (0.48) SMN1; SMN2NPC1RAB9APOLBLMNA
SCHEMBL9049386 0.79 CYP1A2 (0.49) SMN1; SMN2NPC1RAB9APOLBCYP1A2
SCHEMBL16286465 0.79 SMN1; SMN2 (1.00) SMN1; SMN2NPC1RAB9APOLBTDP1
SCHEMBL9050448 0.78 TRPV1 (0.47) SMN1; SMN2NPC1RAB9APOLBLMNA
SCHEMBL7325548 0.76 SMN1; SMN2 (0.45) SMN1; SMN2NPC1RAB9APOLBLMNA
SCHEMBL7327986 0.76 L3MBTL1 (0.47) SMN1; SMN2NPC1RAB9ATDP1LMNA
Fumaric Acid SCHEMBL7334141 0.75 HPGD (0.43) SMN1; SMN2NPC1RAB9ALMNAMAPT
Hydrochloric Acid SCHEMBL9050917 0.75 HTR3A (0.39) ADORA2AADORA1LMNAMAPT
SCHEMBL5897586 0.74 SMN1; SMN2 (0.84) SMN1; SMN2NPC1RAB9APOLBTDP1
SCHEMBL7324842 0.74 KDM4E (0.43) TDP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0381422-B1 Tetrahydrobenzimidazole derivatives YAMANOUCHI PHARMA CO LTD (JP) 1996-10-23 EP disclosed
US-5496942-A 5-HT3-RECEPTOR ANTAGONISTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-03-05 US disclosed
US-5344927-A 5-HT3 antagonist YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1994-09-06 US disclosed
EP-0381422-A1 Tetrahydrobenzimidazole derivatives YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1990-08-08 EP disclosed